SCHEMBL21777464

SCHEMBL21777464

O=C(O)C(NCc1ccc(C(F)(F)F)cc1)C1COC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
EPHX2 P34913 1/20 0.42
PPARG P37231 1/20 0.42
PPARA Q07869 1/20 0.42
FFAR1 O14842 1/20 0.41
P2RX7 Q99572 2/20 0.41
MAPK14 Q16539 1/20 0.39
TEAD1 P28347 1/20 0.39
HIF1A Q16665 1/20 0.39
EPAS1 Q99814 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MAOA P21397 2/20 0.39
KDM1A O60341 1/20 0.39
MAOB P27338 1/20 0.39
MTOR P42345 1/20 0.39
MC4R P32245 1/20 0.38
KCNH2 Q12809 1/20 0.38
TMEM97 Q5BJF2 1/20 0.38
LSS P48449 1/20 0.38
HDAC3 O15379 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21777405 0.86 ALDH1A1 (0.43) ALDH1A1EPHX2PPARGPPARAP2RX7
SCHEMBL21777664 0.85 ITGB3 (0.47) ALDH1A1EPHX2PPARGPPARAFFAR1
SCHEMBL21777494 0.85 ITGB3 (0.47) ALDH1A1EPHX2PPARGPPARAFFAR1
SCHEMBL6235327 0.73 ALDH1A1 (0.58) ALDH1A1EPHX2PPARGPPARAFFAR1
SCHEMBL21789150 0.72 ITGB3 (0.45) ALDH1A1EPHX2PPARGP2RX7TEAD1
SCHEMBL21865730 0.72 ITGB3 (0.45) ALDH1A1EPHX2PPARGP2RX7TEAD1
SCHEMBL11896375 0.70 HTT (0.43) ALDH1A1
SCHEMBL15898200 0.70 HTT (0.40) ALDH1A1MC4R
SCHEMBL17138252 0.69 HPGD (0.46) ALDH1A1FFAR1L3MBTL1MC4R
SCHEMBL19650804 0.69 BCHE (0.52) ALDH1A1EPHX2P2RX7TEAD1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3843842-A1 CARDIAC SARCOMERE INHIBITORS Cytokinetics, Inc. (US) 2021-07-07 EP disclosed
WO-2020047447-A1 CARDIAC SARCOMERE INHIBITORS CYTOKINETICS, INC. (US) 2020-03-05 WO disclosed