SCHEMBL2177875

SCHEMBL2177875

C[C@H](O)[C@@H](N)C(NNCc1ccc(-c2ccccn2)cc1)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 16/20 0.40
CCNE1 P24864 15/20 0.40
CDK5 Q00535 10/20 0.40
CDK9 P50750 2/20 0.39
CDK1 P06493 1/20 0.39
CDK7 P50613 1/20 0.39
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CCNT1 O60563 1/20 0.37
CCNA2 P20248 1/20 0.37
CSNK1A1 P48729 1/20 0.37
GSK3A P49840 1/20 0.37
GSK3B P49841 1/20 0.37
CCNA1 P78396 1/20 0.37
DYRK1A Q13627 1/20 0.37
CDK5R1 Q15078 1/20 0.37
EPHX1 P07099 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3623080 0.76 DPP4 (0.36) CDK2CCNE1CDK5CDK9CDK1
Hydrochloric Acid SCHEMBL3457256 0.76 DPP4 (0.36) CDK2CCNE1CDK5CDK9CDK1
SCHEMBL2179773 0.72 CDK2 (0.46) CDK2CCNE1CDK5CDK9CDK1
SCHEMBL13315147 0.71 CYP2D6 (0.47) CDK2CCNE1CDK5LMNAEPHX1
SCHEMBL13536689 0.71 HCAR2 (0.43) CDK2CCNE1CDK5CDK9CDK1
SCHEMBL5719719 0.70 DPP4 (0.43) CDK2CCNE1CDK5CDK9CDK1
SCHEMBL6895745 0.70 LMNA (0.47) ALDH1A1LMNAMAPK1HTTNPSR1
SCHEMBL6887798 0.70 GAA (0.45) ALDH1A1LMNAMAPK1HTTNPSR1
SCHEMBL893594 0.69 HCAR2 (0.55) LMNAEPHX1CYP2D6EPHX2HIF1A
SCHEMBL12327091 0.68 CCNE1 (0.46) CDK2CCNE1CDK5CDK9CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011080562-A1 NOVEL AZA-PEPTIDES CONTAINING 2,2-DISUBSTITUTED CYCLOBUTYL AND/OR SUBSTITUTED ALKOXY BENZYL DERIVATIVES AS ANTIVIRALS HETERO RESEARCH FOUNDATION (IN) 2011-07-07 WO disclosed
EP-1697348-A1 HIV PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 2006-09-06 EP disclosed
WO-2005061487-A1 HIV PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 2005-07-07 WO disclosed