SCHEMBL2179773

SCHEMBL2179773

CC(O)CCNNCc1ccc(-c2ccccn2)cc1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 19/20 0.46
CCNE1 P24864 17/20 0.46
CDK5 Q00535 11/20 0.46
CDK9 P50750 3/20 0.46
CDK1 P06493 1/20 0.46
CDK7 P50613 1/20 0.46
CCNT1 O60563 2/20 0.44
CCNA2 P20248 2/20 0.44
CSNK1A1 P48729 2/20 0.44
CCNA1 P78396 2/20 0.44
DYRK1A Q13627 2/20 0.44
CDK5R1 Q15078 2/20 0.44
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2175634 0.83 EPHX1 (0.42) CDK2CCNE1CDK5CDK9CCNT1
SCHEMBL13315147 0.77 CYP2D6 (0.47) CDK2CCNE1CDK5
SCHEMBL12327091 0.74 CCNE1 (0.46) CDK2CCNE1CDK5CDK9CDK1
SCHEMBL13536689 0.74 HCAR2 (0.43) CDK2CCNE1CDK5CDK9CDK1
SCHEMBL2237883 0.74 ADRB2 (0.51) CDK2CCNE1CDK5
SCHEMBL16781356 0.74 CXCR4 (0.50) CDK2CCNE1CDK5
SCHEMBL12280795 0.73 CYP2D6 (0.44) CDK2CCNE1CDK5CDK9CDK1
SCHEMBL2179770 0.73 CA12 (0.41) CDK2CCNE1CDK5CDK9CDK1
SCHEMBL2177875 0.72 CDK2 (0.40) CDK2CCNE1CDK5CDK9CDK1
SCHEMBL893594 0.72 HCAR2 (0.55)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011080562-A1 NOVEL AZA-PEPTIDES CONTAINING 2,2-DISUBSTITUTED CYCLOBUTYL AND/OR SUBSTITUTED ALKOXY BENZYL DERIVATIVES AS ANTIVIRALS HETERO RESEARCH FOUNDATION (IN) 2011-07-07 WO disclosed