SCHEMBL21780133

SCHEMBL21780133

C=C(CN)COc1ccc(C(=O)N2Cc3ccc(Cl)cc3C2)cc1F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.39
ENPP2 Q13822 1/20 0.38
ATXN2 Q99700 1/20 0.38
SLC6A9 P48067 1/20 0.38
SLC6A5 Q9Y345 1/20 0.38
TRAP1 Q12931 3/20 0.37
HSP90B1 P14625 2/20 0.37
HPGD P15428 2/20 0.37
USP2 O75604 1/20 0.37
KLKB1 P03952 1/20 0.36
GRM5 P41594 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
HTT P42858 1/20 0.35
MRGPRX4 Q96LA9 1/20 0.35
SLC6A4 P31645 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
TSHR P16473 2/20 0.35
MAPT P10636 2/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21780106 0.84 CPT2 (0.43) NPC1ENPP2ATXN2TRAP1HSP90B1
SCHEMBL21845107 0.73 PARP10 (0.48) NPC1MEN1KMT2AMAPTGAA
SCHEMBL21780048 0.71 AOC2 (0.52) MAOB
SCHEMBL21780093 0.69 HPGD (0.50) NPC1HPGDMEN1KMT2ASMN1; SMN2
SCHEMBL21780098 0.69 HPGD (0.50) NPC1HPGDMEN1KMT2ASMN1; SMN2
SCHEMBL30089453 0.68 MAOB (0.56) ENPP2ATXN2TRAP1HSP90B1HPGD
SCHEMBL21768167 0.68 MAOB (0.56) ENPP2ATXN2TRAP1HSP90B1HPGD
Trifluoroacetic Acid SCHEMBL21768119 0.67 AOC2 (0.48) MAOB
SCHEMBL28901210 0.66 AOC2 (0.42) NPC1ENPP2ATXN2TSHRMAPT
Trifluoroacetic Acid SCHEMBL30089479 0.65 HPGD (0.45) NPC1HPGDMEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3617186-A1 FLUOROALLYLAMINE DERIVATIVE AND USE THEREOF Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. (CN) 2020-03-04 EP disclosed