SCHEMBL21780676

SCHEMBL21780676

CCc1cnc(N2CCNC(=O)C2)nc1C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.49
OPRL1 P41146 3/20 0.49
AOC3 Q16853 1/20 0.41
PDE5A O76074 1/20 0.39
PIK3CA P42336 2/20 0.37
MTOR P42345 1/20 0.37
ADRB1 P08588 1/20 0.36
HPGDS O60760 1/20 0.36
FGFR3 P22607 1/20 0.35
KDR P35968 1/20 0.35
IKBKB O14920 1/20 0.34
PRKCH P24723 1/20 0.34
PRKCE Q02156 1/20 0.34
CCNT1 O60563 1/20 0.34
CDK4 P11802 1/20 0.34
CCND1 P24385 1/20 0.34
CCND3 P30281 1/20 0.34
CDK9 P50750 1/20 0.34
CDK6 Q00534 1/20 0.34
SCN9A Q15858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19145317 0.88 OPRM1 (0.50) OPRM1OPRL1AOC3PDE5APIK3CA
SCHEMBL19105592 0.83 OPRM1 (0.49) OPRM1OPRL1AOC3PDE5APIK3CA
SCHEMBL21768428 0.82 OPRM1 (0.48) OPRM1OPRL1AOC3PDE5APIK3CA
SCHEMBL26342031 0.78 OPRM1 (0.44) OPRM1OPRL1AOC3PDE5APIK3CA
SCHEMBL25075257 0.76 AOC3 (0.44) OPRM1OPRL1AOC3ADRB1HPGDS
SCHEMBL26352347 0.73 AOC3 (0.43) OPRM1OPRL1AOC3PIK3CAMTOR
SCHEMBL22538528 0.72 OPRL1 (0.46) OPRL1KDM4ENR1H2NR1H3
SCHEMBL21780754 0.72 OPRM1 (0.48) OPRM1OPRL1AOC3PIK3CAMTOR
SCHEMBL15415745 0.72 ADRB1 (0.39) OPRM1OPRL1AOC3PIK3CAMTOR
SCHEMBL19117494 0.71 AOC3 (0.49) OPRM1OPRL1AOC3PIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3402781-B1 3-((HETERO-)ARYL)-8-AMINO-2-OXO-1,3-DIAZA-SPIRO-[4.5]-DECANE DERIVATIVES GRUENENTHAL GMBH (DE) 2020-03-04 EP disclosed