SCHEMBL21780689

SCHEMBL21780689

CCCN(CCC)c1cnc(C)cn1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 3/20 0.46
AR P10275 2/20 0.41
DRD2 P14416 1/20 0.37
DRD3 P35462 1/20 0.37
AOC3 Q16853 1/20 0.36
CRHR1 P34998 6/20 0.34
GBA1 P04062 1/20 0.33
HTT P42858 1/20 0.32
MAP3K5 Q99683 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16664161 0.91 HCAR3 (0.44) HCAR3ARDRD2DRD3AOC3
SCHEMBL9924584 0.83 GBA1 (0.48) AOC3CRHR1GBA1
SCHEMBL21769443 0.74 HCAR3 (0.33) HCAR3
SCHEMBL20056973 0.73 HCAR3 (0.57) HCAR3ARDRD2DRD3AOC3
SCHEMBL179289 0.72 AOC3 (0.35) HCAR3AOC3GBA1
SCHEMBL16646632 0.72 HCAR3 (0.44) HCAR3ARDRD2DRD3AOC3
SCHEMBL46324 0.70 MEN1 (0.37)
SCHEMBL2629280 0.69 POLB (0.35) HCAR3GBA1
SCHEMBL2629283 0.69 HRH3 (0.44) HCAR3
SCHEMBL20038496 0.69 CRHR1 (0.42) HCAR3CRHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3402781-B1 3-((HETERO-)ARYL)-8-AMINO-2-OXO-1,3-DIAZA-SPIRO-[4.5]-DECANE DERIVATIVES GRUENENTHAL GMBH (DE) 2020-03-04 EP disclosed