SCHEMBL21781776

SCHEMBL21781776

CNC(CCCNC(N)=O)C(=O)Nc1ccc(CNC(=O)C(Cc2ccccn2)NC(=O)C(C)C(OC)C2CCCN2C)cc1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 1/20 0.38
AKT1 P31749 3/20 0.35
MAPK14 Q16539 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
MAPK1 P28482 1/20 0.34
CYP3A4 P08684 1/20 0.34
MMP3 P08254 4/20 0.33
MMP1 P03956 1/20 0.33
REN P00797 1/20 0.33
USP30 Q70CQ3 1/20 0.33
FKBP4 Q02790 1/20 0.33
NPY1R P25929 1/20 0.33
KDM1A O60341 1/20 0.32
MMP2 P08253 2/20 0.32
GNRHR P30968 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21781988 0.91 KDM1A (0.41) AKT1FKBP4KDM1A
SCHEMBL21782019 0.85 SMN1; SMN2 (0.40) MAPK14SMN1; SMN2MAPK1CYP3A4
SCHEMBL21782055 0.83 FKBP4 (0.39) AKT1MMP3MMP1FKBP4KDM1A
SCHEMBL21781926 0.80 AKT1 (0.42) AKT1
SCHEMBL21782113 0.79 AKT1 (0.41) AKT1CYP3A4KDM1A
SCHEMBL21781982 0.78 AKT1 (0.31) AKT1
SCHEMBL22561364 0.78 KDM1A (0.39) AKT1MMP1USP30FKBP4KDM1A
SCHEMBL21781948 0.77 AKT1 (0.41) AKT1CYP3A4
SCHEMBL22561427 0.77 KLKB1 (0.44) MMP1FKBP4
SCHEMBL21781778 0.76 KLKB1 (0.40) AKT1MMP1FKBP4KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3617221-A1 CYTOTOXIN AND CONJUGATE, USES OF SAME, AND PREPARATION METHOD THEREFOR Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. (CN) 2020-03-04 EP disclosed