SCHEMBL21782113

SCHEMBL21782113

COC(C(C)C(=O)NC(Cc1ccccc1)C(=O)NCc1ccc(NC(=O)C(CCCNC(N)=O)NC(=O)CNC(=O)CCC(=O)N2CCC(C(N)=O)CC2)cc1)C1CCCN1C

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 3/20 0.41
KMT2A Q03164 3/20 0.39
PSMB8 P28062 2/20 0.38
PSMB5 P28074 2/20 0.37
CYP3A4 P08684 1/20 0.37
MEN1 O00255 1/20 0.37
LCK P06239 2/20 0.36
ITGB1 P05556 2/20 0.36
ITGA5 P08648 1/20 0.36
STAT3 P40763 1/20 0.36
ITGA4 P13612 1/20 0.35
KDM1A O60341 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21782075 0.93 AKT1 (0.40) AKT1KMT2APSMB8CYP3A4MEN1
SCHEMBL21781883 0.93 AKT1 (0.40) AKT1KMT2APSMB8PSMB5CYP3A4
SCHEMBL21781948 0.90 AKT1 (0.41) AKT1KMT2APSMB8PSMB5CYP3A4
SCHEMBL21781926 0.89 AKT1 (0.42) AKT1PSMB8PSMB5LCKITGB1
SCHEMBL21781797 0.88 AKT1 (0.39) AKT1KMT2ACYP3A4MEN1LCK
SCHEMBL21782125 0.88 CYP3A4 (0.39) AKT1KMT2ACYP3A4ITGB1ITGA5
SCHEMBL21781939 0.87 AKT1 (0.37) AKT1KMT2APSMB8PSMB5CYP3A4
SCHEMBL21781988 0.86 KDM1A (0.41) AKT1KMT2AMEN1LCKKDM1A
SCHEMBL21781845 0.85 ITGB1 (0.41) AKT1KMT2APSMB8PSMB5MEN1
SCHEMBL21782055 0.79 FKBP4 (0.39) AKT1KMT2AMEN1LCKKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3617221-A1 CYTOTOXIN AND CONJUGATE, USES OF SAME, AND PREPARATION METHOD THEREFOR Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. (CN) 2020-03-04 EP disclosed