SCHEMBL21781883

SCHEMBL21781883

COC(C(C)C(=O)NC(Cc1ccccc1)C(=O)NCc1ccc(NC(=O)C(CCCNC(N)=O)NC(=O)CNC(=O)CCC(=O)N2CCC(C(N)=O)C(C)C2)cc1)C1CCCN1C

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 3/20 0.40
CYP3A4 P08684 1/20 0.36
LCK P06239 2/20 0.35
PSMB8 P28062 2/20 0.35
PSMB5 P28074 1/20 0.35
ITGB1 P05556 1/20 0.35
ITGA5 P08648 1/20 0.35
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
F2R P25116 2/20 0.34
STAT3 P40763 1/20 0.34
NMUR2 Q9GZQ4 1/20 0.34
NMUR1 Q9HB89 1/20 0.34
OPRK1 P41145 1/20 0.34
KLKB1 P03952 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21782113 0.93 AKT1 (0.41) AKT1CYP3A4LCKPSMB8PSMB5
SCHEMBL21782075 0.89 AKT1 (0.40) AKT1CYP3A4LCKPSMB8ITGB1
SCHEMBL21781926 0.88 AKT1 (0.42) AKT1LCKPSMB8PSMB5ITGB1
SCHEMBL21782124 0.86 ITGB1 (0.38) AKT1LCKPSMB8PSMB5ITGB1
SCHEMBL21781948 0.86 AKT1 (0.41) AKT1CYP3A4LCKPSMB8PSMB5
SCHEMBL21781988 0.85 KDM1A (0.41) AKT1LCKKLKB1MEN1KMT2A
SCHEMBL21782125 0.84 CYP3A4 (0.39) AKT1CYP3A4ITGB1ITGA5OPRM1
SCHEMBL21781797 0.83 AKT1 (0.39) AKT1CYP3A4LCKITGB1ITGA5
SCHEMBL21781845 0.81 ITGB1 (0.41) AKT1LCKPSMB8PSMB5ITGB1
SCHEMBL21782000 0.79 ITGB1 (0.34) ITGB1ITGA5KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3617221-A1 CYTOTOXIN AND CONJUGATE, USES OF SAME, AND PREPARATION METHOD THEREFOR Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. (CN) 2020-03-04 EP disclosed