SCHEMBL21782124

SCHEMBL21782124

CNCCCC(NC(=O)CNC(=O)CCC(=O)N1CCC(C(N)=O)C(C)C1)C(=O)Nc1ccc(CNC(=O)C(Cc2ccccc2)NC(=O)C(C)C(OC)C2CCCN2)cc1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 2/20 0.38
ITGA5 P08648 1/20 0.38
AKT1 P31749 3/20 0.37
PSMB8 P28062 2/20 0.34
PSMB5 P28074 1/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
LCK P06239 2/20 0.33
KLKB1 P03952 1/20 0.33
OPRK1 P41145 1/20 0.33
ITGA4 P13612 1/20 0.33
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
HRH1 P35367 1/20 0.32
KDM1A O60341 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21781883 0.86 AKT1 (0.40) ITGB1ITGA5AKT1PSMB8PSMB5
SCHEMBL21782113 0.79 AKT1 (0.41) ITGB1ITGA5AKT1PSMB8PSMB5
SCHEMBL21781845 0.76 ITGB1 (0.41) ITGB1ITGA5AKT1PSMB8PSMB5
SCHEMBL21782075 0.75 AKT1 (0.40) ITGB1ITGA5AKT1PSMB8KMT2A
SCHEMBL21781926 0.74 AKT1 (0.42) ITGB1ITGA5AKT1PSMB8PSMB5
SCHEMBL21782000 0.73 ITGB1 (0.34) ITGB1ITGA5KMT2AITGA4
SCHEMBL21782121 0.73 CYP3A4 (0.43) ITGB1ITGA5AKT1PSMB8PSMB5
SCHEMBL21781948 0.72 AKT1 (0.41) ITGB1ITGA5AKT1PSMB8PSMB5
SCHEMBL21781988 0.71 KDM1A (0.41) AKT1KMT2AMEN1LCKKLKB1
SCHEMBL22561364 0.70 KDM1A (0.39) ITGB1ITGA5AKT1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3617221-A1 CYTOTOXIN AND CONJUGATE, USES OF SAME, AND PREPARATION METHOD THEREFOR Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. (CN) 2020-03-04 EP disclosed