SCHEMBL21782018

SCHEMBL21782018

COC(C(C)C(=O)NC(Cc1ccccc1)C(=O)NCc1ccc(NC(=O)C(CCCNC(N)=O)NC(=O)CNC(=O)CCCN2CCC(C(N)=O)CC2C(F)(F)F)cc1)C1CCCN1C=O

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 3/20 0.37
ITGB1 P05556 1/20 0.34
ITGA5 P08648 1/20 0.34
CYP3A4 P08684 1/20 0.34
QRFPR Q96P65 2/20 0.33
LCK P06239 2/20 0.33
KLKB1 P03952 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
MMP7 P09237 2/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
NMUR2 Q9GZQ4 1/20 0.32
NMUR1 Q9HB89 1/20 0.32
OPRL1 P41146 1/20 0.32
HRH1 P35367 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21781797 0.94 AKT1 (0.39) AKT1ITGB1ITGA5CYP3A4LCK
SCHEMBL21781814 0.87 AKT1 (0.31) AKT1ITGB1ITGA5
SCHEMBL21781887 0.86
SCHEMBL21782058 0.86 CYP3A4 (0.44) AKT1CYP3A4OPRD1
SCHEMBL21781807 0.84 CYP3A4 (0.31) AKT1ITGB1CYP3A4
SCHEMBL21781939 0.83 AKT1 (0.37) AKT1ITGB1ITGA5CYP3A4LCK
SCHEMBL21782113 0.82 AKT1 (0.41) AKT1ITGB1ITGA5CYP3A4LCK
SCHEMBL21782075 0.82 AKT1 (0.40) AKT1ITGB1ITGA5CYP3A4LCK
SCHEMBL21781926 0.81 AKT1 (0.42) AKT1ITGB1ITGA5LCKKLKB1
SCHEMBL21782071 0.81 ITGB1 (0.34) AKT1ITGB1ITGA5MMP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3617221-A1 CYTOTOXIN AND CONJUGATE, USES OF SAME, AND PREPARATION METHOD THEREFOR Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. (CN) 2020-03-04 EP disclosed