SCHEMBL21783687

SCHEMBL21783687

CNc1cccc2ccncc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNF P01375 2/20 0.49
HDAC6 Q9UBN7 1/20 0.46
RORC P51449 1/20 0.42
AOC1 P19801 2/20 0.42
AOC3 Q16853 2/20 0.42
TRPV1 Q8NER1 1/20 0.41
LMNA P02545 2/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
ROCK2 O75116 1/20 0.41
ROCK1 Q13464 1/20 0.41
CCNE1 P24864 1/20 0.40
CDK2 P24941 1/20 0.40
CDK5 Q00535 1/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2D6 P10635 2/20 0.40
CYP1A2 P05177 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1735616 0.85 ROCK2 (0.55) LMNAALDH1A1MAPTKMT2ASMN1; SMN2
SCHEMBL4528495 0.81 KEAP1 (0.65) RORC
SCHEMBL2481375 0.81 TNF (0.49) TNFHDAC6TRPV1LMNAALDH1A1
SCHEMBL2622216 0.80 LATS1 (0.46) TNFHDAC6RORCTRPV1LMNA
SCHEMBL30645377 0.78 MEN1 (0.53) HDAC6TRPV1ALDH1A1MAPTKMT2A
SCHEMBL9651248 0.78 MEN1 (0.53) HDAC6TRPV1ALDH1A1MAPTKMT2A
SCHEMBL30600745 0.75 TRPV1 (0.52) TNFHDAC6TRPV1ALDH1A1MAPT
SCHEMBL49308 0.74 KEAP1 (0.61) LMNAALDH1A1CYP3A4CYP2D6CYP1A2
SCHEMBL17737617 0.74 RECQL (0.69) ALDH1A1MAPTKMT2AALOX12
SCHEMBL2321594 0.74 KDM4E (0.67) TNFHDAC6TRPV1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020047208-A1 INHIBITORS OF (ALPHA-V)(BETA-6) INTEGRIN MORPHIC THERAPEUTIC, INC. (US) 2020-03-05 WO disclosed
CN-110669058-A Tricyclic quinolone carboxylic acid and preparation method thereof 江西农业大学 2020-01-10 CN disclosed