SCHEMBL21788050

SCHEMBL21788050

COC(=O)c1cc(C(C)=O)oc1C(C)c1ccc(C)cc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 13/20 0.48
POLB P06746 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CA12 O43570 2/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA7 P43166 2/20 0.38
CA9 Q16790 2/20 0.38
CA14 Q9ULX7 2/20 0.38
PDK2 Q15119 1/20 0.38
PDK4 Q16654 1/20 0.38
GAA P10253 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ALDH1A1 P00352 1/20 0.37
BRD2 P25440 1/20 0.37
BRD3 Q15059 1/20 0.37
BRDT Q58F21 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24006927 0.87 BRD4 (0.63) BRD4POLBBRD2BRD3BRDT
SCHEMBL21787800 0.77 BRD4 (0.68) BRD4BRD2BRD3BRDT
SCHEMBL21787793 0.76 BRD4 (0.40) BRD4POLBGAAL3MBTL1ALDH1A1
SCHEMBL21787790 0.75 BRD4 (0.70) BRD4POLBGAABRD2BRD3
SCHEMBL21787789 0.75 BRD4 (0.70) BRD4POLBGAABRD2BRD3
SCHEMBL21776776 0.75 BRD4 (0.67) BRD4TDP1L3MBTL1ALDH1A1BRD2
SCHEMBL12494900 0.72 ALDH1A1 (0.44) POLBGAAL3MBTL1ALDH1A1
SCHEMBL24006876 0.72 BRD4 (0.48) BRD4BRD2BRD3BRDT
SCHEMBL21787943 0.70 BRD4 (0.45) BRD4TDP1CA12CA1CA2
SCHEMBL21787719 0.69 BRD4 (0.66) BRD4POLBALDH1A1BRD2BRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020043821-A1 FURAN DERIVATIVES AS BROMODOMAIN INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED (GB) 2020-03-05 WO disclosed