SCHEMBL21787793

SCHEMBL21787793

CC(=O)c1cc(C=O)c(C(C)c2ccc(C)cc2)o1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 6/20 0.40
TYR P14679 1/20 0.39
ERN1 O75460 1/20 0.38
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 2/20 0.37
GAA P10253 2/20 0.37
HSD17B10 Q99714 2/20 0.37
LMNA P02545 1/20 0.37
GLA P06280 1/20 0.37
HPGD P15428 1/20 0.37
CASP1 P29466 1/20 0.37
BRCA1 P38398 1/20 0.37
CASP7 P55210 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
STAT3 P40763 3/20 0.35
MEN1 O00255 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
ALOX12 P18054 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21788050 0.76 BRD4 (0.48) BRD4ALDH1A1GAAPOLBL3MBTL1
SCHEMBL27261858 0.70 ERN1 (0.38) TYRERN1ALDH1A1KDM4EGAA
SCHEMBL21787800 0.69 BRD4 (0.68) BRD4LMNAGLAHPGDSMN1; SMN2
SCHEMBL21776776 0.66 BRD4 (0.67) BRD4ALDH1A1HPGDMEN1MAPT
SCHEMBL822908 0.63 ESR1 (0.80) TYRALDH1A1KDM4EGAAHSD17B10
SCHEMBL24006927 0.63 BRD4 (0.63) BRD4POLB
SCHEMBL21787802 0.63 TAS1R3 (0.44) ALDH1A1GAALMNAHPGDSMN1; SMN2
SCHEMBL2681029 0.63 CYP2A6 (0.70) TYRALDH1A1KDM4EHSD17B10HPGD
SCHEMBL17399576 0.62 TYR (0.69) TYRERN1KDM4EMEN1POLB
P-Cymene SCHEMBL28761802 0.61 TRIM24 (0.60) TYRERN1ALDH1A1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020043821-A1 FURAN DERIVATIVES AS BROMODOMAIN INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED (GB) 2020-03-05 WO disclosed