SCHEMBL21790245

SCHEMBL21790245

COCc1cccc([C@@H](CN)C(=O)Nc2ccc3cnccc3c2)c1

nearest known ligand 0.79

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 20/20 0.79
ROCK1 Q13464 2/20 0.71
MYLK4 Q86YV6 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21790249 1.00 ROCK2 (0.79) ROCK2ROCK1MYLK4
SCHEMBL21790292 0.91 ROCK2 (0.76) ROCK2ROCK1MYLK4
SCHEMBL21790286 0.91 ROCK2 (0.76) ROCK2ROCK1MYLK4
SCHEMBL21795453 0.89 ROCK2 (0.80) ROCK2ROCK1MYLK4
SCHEMBL21790244 0.89 ROCK2 (0.80) ROCK2ROCK1MYLK4
SCHEMBL23633797 0.89 ROCK2 (0.73) ROCK2ROCK1MYLK4
SCHEMBL19932282 0.89 ROCK2 (0.76) ROCK2ROCK1MYLK4
SCHEMBL23866454 0.88 ROCK2 (0.72) ROCK2ROCK1
SCHEMBL19886640 0.87 ROCK2 (1.00) ROCK2ROCK1
SCHEMBL28404271 0.87 ROCK2 (0.73) ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020047496-A1 ISOQUINOLINE-STEROID CONJUGATES AND USES THEREOF AERIE PHARMACEUTICALS, INC. (US) 2020-03-05 WO disclosed