SCHEMBL2179240

SCHEMBL2179240

NC(=O)Cc1cc(Cl)nc(NCc2ccc3ncccc3c2)c1[N+](=O)[O-]

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.41
HDAC3 O15379 2/20 0.40
HDAC6 Q9UBN7 1/20 0.40
KDR P35968 11/20 0.39
FLT1 P17948 1/20 0.38
NPC1 O15118 1/20 0.37
MAPT P10636 1/20 0.36
PKM P14618 1/20 0.36
GLS O94925 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13571271 0.85 HDAC3 (0.45) ALOX5HDAC3HDAC6KDRFLT1
SCHEMBL2177207 0.84 MAPT (0.42) ALOX5HDAC3HDAC6KDRNPC1
SCHEMBL2178270 0.82 ALOX5 (0.43) ALOX5HDAC3HDAC6KDRFLT1
SCHEMBL2175935 0.82 ALOX5 (0.43) ALOX5HDAC3HDAC6KDRFLT1
SCHEMBL2195228 0.81 ALOX5 (0.42) ALOX5HDAC3HDAC6KDRFLT1
SCHEMBL12544010 0.78 ALOX5 (0.40) ALOX5HDAC3HDAC6KDRFLT1
SCHEMBL30779384 0.78 ALOX5 (0.40) ALOX5HDAC3HDAC6KDRFLT1
SCHEMBL1330877 0.77 MAPT (0.49) ALOX5HDAC6KDRNPC1MAPT
SCHEMBL3394316 0.72 PIN1 (0.48) HDAC6KDRNPC1
SCHEMBL12544218 0.71 HDAC3 (0.47) ALOX5HDAC3HDAC6KDRFLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2519524-A1 CERTAIN TRIAZOLOPYRIDINES AND TRIAZOLOPYRAZINES, COMPOSITIONS THEREOF AND METHODS OF USE THEREFOR Hutchison Medipharma Limited (CN) 2012-11-07 EP disclosed
WO-2011079804-A1 CERTAIN TRIAZOLOPYRIDINES AND TRIAZOLOPYRAZINES, COMPOSITIONS THEREOF AND METHODS OF USE THEREFOR HUTCHISON MEDIPHARMA LIMITED (CN) 2011-07-07 WO disclosed