SCHEMBL21793293

SCHEMBL21793293

COc1cc2nccc(Oc3ccc(N=O)cc3F)c2c2c1OCCO2

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDR P35968 10/20 0.61
RET P07949 7/20 0.61
MET P08581 3/20 0.49
EGFR P00533 1/20 0.43
AXL P30530 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21750981 0.85 KDR (0.61) KDRRETMETEGFRAXL
SCHEMBL21265686 0.83 KDR (0.69) KDRRETMETEGFRAXL
SCHEMBL21246953 0.83 KDR (0.59) KDRRETMETEGFR
SCHEMBL23749325 0.79 KDR (0.54) KDRRETMETEGFRAXL
SCHEMBL23749306 0.78 KDR (0.58) KDRRETMETEGFR
SCHEMBL13955465 0.78 FGFR2 (0.58) KDRMETAXL
SCHEMBL21793294 0.77 KDR (0.68) KDRRETMET
SCHEMBL23749294 0.77 KDR (0.56) KDRRETMETEGFR
SCHEMBL21751008 0.76 RET (0.61) KDRRETMETEGFR
SCHEMBL30664551 0.76 RET (0.61) KDRRETMETEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020042972-A1 UREA-SUBSTITUTED AROMATIC RING-LINKED DIOXANE AND QUINAZOLINE OR QUINOLINE COMPOUND, COMPOSITION AND APPLICATION THEREOF 北京赛特明强医药科技有限公司 2020-03-05 WO disclosed