SCHEMBL21793294

SCHEMBL21793294

COc1cc2nccc(Oc3ccc(NC(=O)Oc4ccccc4)cc3F)c2c2c1OCCO2

nearest known ligand 0.68

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDR P35968 8/20 0.68
RET P07949 5/20 0.68
MET P08581 7/20 0.55
KIT P10721 1/20 0.54
PDGFRA P16234 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4298086 0.83 PDGFRA (0.77) KDRMETKITPDGFRA
SCHEMBL21265686 0.83 KDR (0.69) KDRRETMETPDGFRA
SCHEMBL21792996 0.81 RET (0.64) KDRRETMETKITPDGFRA
SCHEMBL21265684 0.81 MET (0.81) KDRRETMETKITPDGFRA
SCHEMBL22821317 0.81 KDR (1.00) KDRRET
SCHEMBL21793056 0.79 RET (0.74) KDRRETMETPDGFRA
SCHEMBL21262599 0.79 KDR (1.00) KDRRET
SCHEMBL21792906 0.79 RET (0.73) KDRRETMETPDGFRA
SCHEMBL30664577 0.79 KDR (1.00) KDRRET
SCHEMBL21793293 0.77 KDR (0.61) KDRRETMET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020042972-A1 UREA-SUBSTITUTED AROMATIC RING-LINKED DIOXANE AND QUINAZOLINE OR QUINOLINE COMPOUND, COMPOSITION AND APPLICATION THEREOF 北京赛特明强医药科技有限公司 2020-03-05 WO disclosed