SCHEMBL21795314

SCHEMBL21795314

O=CC1CCN(c2ccc(C(F)(F)F)c3nccnc23)C1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RBP4 P02753 9/20 0.36
TTR P02766 6/20 0.36
NCF1 P14598 1/20 0.35
NOTUM Q6P988 3/20 0.34
AR P10275 1/20 0.34
PDE3B Q13370 2/20 0.34
PDE3A Q14432 2/20 0.34
CYP2C19 P33261 1/20 0.34
PIK3CA P42336 1/20 0.34
RPS6KB1 P23443 2/20 0.33
AKT1 P31749 1/20 0.33
CYP8B1 Q9UNU6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21795312 0.82 AR (0.42) NCF1NOTUMARPDE3BPDE3A
SCHEMBL23760701 0.82 AR (0.42) NCF1NOTUMARPDE3BPDE3A
SCHEMBL23760683 0.81 MAP4K4 (0.42) NCF1NOTUMARPDE3BPDE3A
SCHEMBL23369720 0.78 NCF1 (0.52) NCF1RPS6KB1
SCHEMBL18991731 0.77 KDM4E (0.49) NOTUMPDE3BPDE3A
SCHEMBL30571038 0.76 PIM2 (0.46) CYP2C19PIK3CA
SCHEMBL28662001 0.76 PIM2 (0.46) CYP2C19PIK3CA
SCHEMBL23760669 0.76 NOTUM (0.39) RBP4NCF1NOTUMARPDE3B
SCHEMBL31648090 0.72 ACACB (0.47) AR
Hydrochloric Acid SCHEMBL31648142 0.71 ACACB (0.46) AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020043271-A1 NOVEL PYRROLIDINYL AMIDE COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE DISEASE F. HOFFMANN-LA ROCHE AG (CH) 2020-03-05 WO disclosed