SCHEMBL2179770

SCHEMBL2179770

CC(O)CCN(N)Cc1ccc(-c2ccccn2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 6/20 0.41
CA1 P00915 6/20 0.41
CA2 P00918 6/20 0.41
CA5A P35218 6/20 0.41
CA9 Q16790 6/20 0.41
CA5B Q9Y2D0 6/20 0.41
CDK2 P24941 6/20 0.41
CCNE1 P24864 5/20 0.41
CDK5 Q00535 5/20 0.41
CDK9 P50750 2/20 0.41
CDK1 P06493 1/20 0.41
CDK7 P50613 1/20 0.41
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP19A1 P11511 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
DPP4 P27487 1/20 0.37
SLC6A9 P48067 1/20 0.37
NR1I2 O75469 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2179765 0.80 CYP1A2 (0.42) CA12CA1CA2CA5ACA9
SCHEMBL8103923 0.78 CCNE1 (0.40) CA12CA1CA2CA5ACA9
SCHEMBL12327804 0.77 HCAR2 (0.40) CA12CA1CA2CA9NR1I2
SCHEMBL19112092 0.76 CYP1A2 (0.45) CA12CA1CA2CA5ACA9
SCHEMBL2177873 0.73 UGT1A1 (0.43) DPP4NR1I2NMBRGRPRBRS3
SCHEMBL8152590 0.73 UGT1A1 (0.43) DPP4NR1I2NMBRGRPRBRS3
SCHEMBL3393562 0.73 UGT1A1 (0.43) DPP4NR1I2NMBRGRPRBRS3
SCHEMBL2179773 0.73 CDK2 (0.46) CDK2CCNE1CDK5CDK9CDK1
SCHEMBL19112162 0.73 TAAR1 (0.58) CA12CA1CA2CA5ACA9
Hydrochloric Acid SCHEMBL1300940 0.72 UGT1A1 (0.43) DPP4NR1I2NMBRGRPRBRS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011080562-A1 NOVEL AZA-PEPTIDES CONTAINING 2,2-DISUBSTITUTED CYCLOBUTYL AND/OR SUBSTITUTED ALKOXY BENZYL DERIVATIVES AS ANTIVIRALS HETERO RESEARCH FOUNDATION (IN) 2011-07-07 WO disclosed