SCHEMBL21806003

SCHEMBL21806003

COC(=O)[C@@H](O)CN1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.45
USP2 O75604 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
ALDH1A1 P00352 3/20 0.43
HTT P42858 2/20 0.42
CHRM2 P08172 1/20 0.42
CHRM4 P08173 1/20 0.42
CHRM1 P11229 1/20 0.42
CHRM3 P20309 1/20 0.42
NPC1 O15118 1/20 0.42
MAPT P10636 1/20 0.42
MAPK1 P28482 1/20 0.42
RAB9A P51151 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
EPHX2 P34913 1/20 0.41
EPHX1 P07099 1/20 0.40
KDM4E B2RXH2 1/20 0.39
NR1H2 P55055 1/20 0.39
HPGD P15428 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24027253 1.00 ABCB1 (0.45) ABCB1USP2SMN1; SMN2ALDH1A1HTT
SCHEMBL2529177 0.85 ALDH1A1 (0.48) ABCB1USP2SMN1; SMN2ALDH1A1HTT
SCHEMBL2529176 0.85 ALDH1A1 (0.48) ABCB1USP2SMN1; SMN2ALDH1A1HTT
SCHEMBL5859962 0.84 USP2 (0.43) ABCB1USP2SMN1; SMN2ALDH1A1HTT
SCHEMBL27385307 0.84 USP2 (0.43) ABCB1USP2SMN1; SMN2ALDH1A1HTT
SCHEMBL21806029 0.84 ABCB1 (0.46) ABCB1USP2SMN1; SMN2ALDH1A1HTT
SCHEMBL24027198 0.84 ABCB1 (0.46) ABCB1USP2SMN1; SMN2ALDH1A1HTT
SCHEMBL29223471 0.83 USP2 (0.50) ABCB1USP2SMN1; SMN2ALDH1A1HTT
SCHEMBL16825817 0.81 USP2 (0.49) ABCB1USP2SMN1; SMN2ALDH1A1HTT
SCHEMBL20232006 0.81 USP2 (0.49) ABCB1USP2SMN1; SMN2ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3853212-A1 ISOXAZOLE CARBOXAMIDE COMPOUNDS AND USES THEREOF Novartis AG (CH) 2021-07-28 EP disclosed
WO-2020058913-A1 ISOXAZOLE CARBOXAMIDE COMPOUNDS AND USES THEREOF NOVARTIS AG (CH) 2020-03-26 WO disclosed