SCHEMBL21807341

SCHEMBL21807341

O=c1c(Cl)c(N2CCc3c(CCc4ccc(F)cc4C(F)(F)F)ncnc3C2)cnn1C1CCCCO1

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPC5 Q9UL62 15/20 0.45
TRPC4 Q9UBN4 2/20 0.45
P2RX3 P56373 3/20 0.32
P2RX2 Q9UBL9 3/20 0.32
AR P10275 1/20 0.32
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29090320 0.84 TRPC5 (0.46) TRPC5TRPC4AR
SCHEMBL29329165 0.84 TRPC5 (0.47) TRPC5TRPC4KMT2A
SCHEMBL21807248 0.84 TRPC5 (0.65) TRPC5TRPC4
SCHEMBL29329169 0.83 TRPC5 (0.45) TRPC5TRPC4P2RX3P2RX2AR
SCHEMBL21807320 0.83 TRPC5 (0.44) TRPC5TRPC4ARKMT2A
SCHEMBL21807339 0.83 TRPC5 (0.46) TRPC5TRPC4
SCHEMBL31058992 0.83 TRPC5 (0.46) TRPC5TRPC4
SCHEMBL22002665 0.83 TRPC5 (0.46) TRPC5TRPC4
SCHEMBL29329276 0.83 TRPC5 (0.44) TRPC5TRPC4AR
SCHEMBL20831591 0.82 TRPC5 (0.41) TRPC5TRPC4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3941475-A1 PYRIDAZINONES AND METHODS OF USE THEREOF Goldfinch Bio, Inc. (US) 2022-01-26 EP disclosed
EP-3852533-A1 PYRIDAZINONES AND METHODS OF USE THEREOF Goldfinch Bio, Inc. (US) 2021-07-28 EP disclosed
WO-2020191056-A1 PYRIDAZINONES AND METHODS OF USE THEREOF GOLDFINCH BIO, INC. (US) 2020-09-24 WO disclosed
WO-2020061162-A1 PYRIDAZINONES AND METHODS OF USE THEREOF GOLDFINCH BIO, INC. (US) 2020-03-26 WO disclosed