SCHEMBL21811816

SCHEMBL21811816

O=C(O)C1CC(OCCOCc2ccccc2)C1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
LIPG Q9Y5X9 1/20 0.43
ALDH1A1 P00352 2/20 0.43
GAA P10253 1/20 0.43
EPHX2 P34913 2/20 0.42
AGTR2 P50052 5/20 0.42
TSHR P16473 1/20 0.41
S1PR5 Q9H228 1/20 0.41
HTT P42858 1/20 0.40
PDE4D Q08499 1/20 0.40
TEAD3 Q99594 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7988899 0.87 ALDH1A1 (0.51) SMN1; SMN2NPC1RAB9ALIPGALDH1A1
SCHEMBL21801247 0.86 ALDH1A1 (0.42) SMN1; SMN2NPC1RAB9ALIPGALDH1A1
SCHEMBL871908 0.85 NPC1 (0.49) SMN1; SMN2NPC1RAB9AALDH1A1GAA
SCHEMBL8347290 0.85 NPC1 (0.49) SMN1; SMN2NPC1RAB9AALDH1A1GAA
SCHEMBL582677 0.85 NPC1 (0.49) SMN1; SMN2NPC1RAB9AALDH1A1GAA
SCHEMBL29224959 0.83 S1PR5 (0.46) SMN1; SMN2NPC1RAB9AALDH1A1GAA
SCHEMBL21801225 0.83 L3MBTL1 (0.45) RAB9ALIPGGAAEPHX2
SCHEMBL21801224 0.83 L3MBTL1 (0.45) RAB9ALIPGGAAEPHX2
SCHEMBL20132896 0.81 PDE4D (0.44) SMN1; SMN2LIPGALDH1A1EPHX2TSHR
SCHEMBL21812039 0.81 L3MBTL1 (0.51) ALDH1A1EPHX2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3860984-A1 FLAVONE DERIVATIVES FOR THE TREATMENT AND PROPHYLAXIS OF HEPATITIS B VIRUS DISEASE F. Hoffmann-La Roche AG (CH) 2021-08-11 EP disclosed
EP-3849966-A1 FLAVONE COMPOUNDS FOR THE TREATMENT AND PROPHYLAXIS OF HEPATITIS B VIRUS DISEASE F. Hoffmann-La Roche AG (CH) 2021-07-21 EP disclosed
WO-2021063856-A1 SUBSTITUTED 3,4-DIHYDROQUINAZOLINE FOR THE TREATMENT AND PROPHYLAXIS OF HEPATITIS B VIRUS INFECTION F. HOFFMANN-LA ROCHE AG (CH) 2021-04-08 WO disclosed
CN-112601743-A Flavone compounds for treating and preventing hepatitis B virus diseases 豪夫迈·罗氏有限公司 2021-04-02 CN disclosed
WO-2020070088-A1 FLAVONE DERIVATIVES FOR THE TREATMENT AND PROPHYLAXIS OF HEPATITIS B VIRUS DISEASE F. HOFFMANN-LA ROCHE AG (CH) 2020-04-09 WO disclosed
WO-2020053249-A1 FLAVONE COMPOUNDS FOR THE TREATMENT AND PROPHYLAXIS OF HEPATITIS B VIRUS DISEASE F. HOFFMANN-LA ROCHE AG (CH) 2020-03-19 WO disclosed