SCHEMBL2183228

SCHEMBL2183228

CCCOCCOC(=O)C(C)=C[Si](O[Si](C)(C)C)(O[Si](C)(C)C)O[Si](C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.37
ALDH1A1 P00352 3/20 0.33
TSHR P16473 3/20 0.33
TP53 P04637 2/20 0.33
HIF1A Q16665 2/20 0.33
HSD17B10 Q99714 1/20 0.33
HCAR2 Q8TDS4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL525364 0.91 HCAR2 (0.38) THRBALDH1A1TSHRHCAR2
SCHEMBL9354366 0.80
SCHEMBL28359357 0.78 HCAR2 (0.38) THRBALDH1A1TSHRHCAR2
SCHEMBL7777475 0.77 THRB (0.46) THRBALDH1A1TSHRTP53HIF1A
SCHEMBL27924395 0.76 HCAR2 (0.33) TSHRHCAR2
SCHEMBL146699 0.74 HCAR2 (0.36) THRBALDH1A1TSHRHCAR2
SCHEMBL30018944 0.74 HCAR2 (0.36) THRBALDH1A1TSHRHCAR2
SCHEMBL4642491 0.73 HCAR2 (0.38) THRBALDH1A1TSHRHCAR2
SCHEMBL1155539 0.73 TSHR (0.33) TSHR
SCHEMBL425966 0.72 HCAR2 (0.35) THRBALDH1A1TSHRHSD17B10HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102675561-B silicone hydrogel with high water content FAR EASTERN NEW CENTURY CORPORATION (CN) 2014-10-22 CN claimed
CN-102675658-A Method for preparing polysiloxane hydrogel with high moisture content FAR EASTERN NEW CENTURY CORP 2012-09-19 CN claimed
CN-102675561-A Silicone hydrogel with high water content FAR EASTERN NEW CENTURY CORP 2012-09-19 CN claimed
CN-102464744-A Chlorinated polymers that enhance wettability of silicone hydrogels, silicone hydrogels comprising the same, and ophthalmic articles made therefrom FAR EASTERN NEW CENTURY CORP 2012-05-23 CN claimed
US-20120115979-A1 CHLORINATED POLYMER ENHANCING WETTABILITY OF SILICONE HYDROGEL, SILICONE HYDROGEL COMPRISING THE SAME AND OCULAR ARTICLE MADE THEREFROM FAR EASTERN NEW CENTURY CORPORATION (TW) 2012-05-10 US claimed
US-20110166248-A1 COPOLYMER FOR ENHANCING THE wETTABILITY OF SILICONE HYDROGEL, SILICONE HYDROGEL COMPOSITION COMPRISING THE SAME AND OCULAR ARTICLE MADE THEREFROM FAR EASTERN NEW CENTURY CORPORATION 2011-07-07 US claimed
CN-102675561-B silicone hydrogel with high water content FAR EASTERN NEW CENTURY CORPORATION (CN) 2014-10-22 CN disclosed
US-8492513-B2 Method for enhancing water content of silicone hydrogel contact lens FAR EASTERN NEW CENTURY CORPORATION (TW) 2013-07-23 US disclosed
CN-102675658-A Method for preparing polysiloxane hydrogel with high moisture content FAR EASTERN NEW CENTURY CORP 2012-09-19 CN disclosed
CN-102675561-A Silicone hydrogel with high water content FAR EASTERN NEW CENTURY CORP 2012-09-19 CN disclosed
US-20120214899-A1 METHOD FOR ENHANCING WATER CONTENT OF SILICONE HYDROGEL CONTACT LENS FAR EASTERN NEW CENTURY CORPORATION (TW) 2012-08-23 US disclosed
CN-102464744-A Chlorinated polymers that enhance wettability of silicone hydrogels, silicone hydrogels comprising the same, and ophthalmic articles made therefrom FAR EASTERN NEW CENTURY CORP 2012-05-23 CN disclosed
US-20120115979-A1 CHLORINATED POLYMER ENHANCING WETTABILITY OF SILICONE HYDROGEL, SILICONE HYDROGEL COMPRISING THE SAME AND OCULAR ARTICLE MADE THEREFROM FAR EASTERN NEW CENTURY CORPORATION (TW) 2012-05-10 US disclosed
US-20110166248-A1 COPOLYMER FOR ENHANCING THE wETTABILITY OF SILICONE HYDROGEL, SILICONE HYDROGEL COMPOSITION COMPRISING THE SAME AND OCULAR ARTICLE MADE THEREFROM FAR EASTERN NEW CENTURY CORPORATION 2011-07-07 US disclosed