SCHEMBL21845810

SCHEMBL21845810

CC(=O)[C@@H]1C[C@H]1c1ccc(S(C)(=O)=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.44
SCN3A Q9NY46 1/20 0.43
ENPP2 Q13822 2/20 0.42
KDM1A O60341 1/20 0.42
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
RIPK1 Q13546 1/20 0.40
FFAR1 O14842 2/20 0.40
PTGS2 P35354 3/20 0.39
TGM2 P21980 1/20 0.39
KMT2A Q03164 1/20 0.39
NAMPT P43490 1/20 0.38
HDAC4 P56524 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18231177 1.00 SLC6A4 (0.44) SLC6A4SCN3AENPP2KDM1AMAOA
SCHEMBL21845698 1.00 SLC6A4 (0.44) SLC6A4SCN3AENPP2KDM1AMAOA
SCHEMBL15212214 0.86 FFAR1 (0.54) SLC6A4SCN3AENPP2KDM1AMAOA
SCHEMBL23107750 0.85 CHRNA7 (0.47) SCN3ACYP3A4CYP2C9ALDH1A1CYP1A2
SCHEMBL19378449 0.85 CHRNA7 (0.47) SCN3ACYP3A4CYP2C9ALDH1A1CYP1A2
SCHEMBL19683268 0.80 ENPP2 (0.45) SLC6A4ENPP2KDM1AMAOAMAOB
SCHEMBL13527048 0.80 ENPP2 (0.45) SLC6A4ENPP2KDM1AMAOAMAOB
SCHEMBL15212285 0.79 SLC6A4 (0.44) SLC6A4KDM1AMAOAMAOBCYP3A4
SCHEMBL21845792 0.78 ALDH1A1 (0.64) SLC6A4CYP3A4CYP2C9ALDH1A1CYP1A2
SCHEMBL799523 0.78 ALDH1A1 (0.64) SLC6A4CYP3A4CYP2C9ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020056345-A1 ARYL CYCLOPROPYL-AMINO-ISOQUINOLINYL AMIDE COMPOUNDS AERIE PHARMACEUTICALS, INC. (US) 2020-03-19 WO disclosed