SCHEMBL21851206

SCHEMBL21851206

C1=C\C=C/C=C\C(NNc2ccccccccc2)=C/C=C\C=C/1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 4/20 0.52
ALDH1A1 P00352 4/20 0.52
CTSD P07339 1/20 0.52
HSD17B10 Q99714 2/20 0.35
TSHR P16473 3/20 0.33
PTGS2 P35354 3/20 0.33
CYP3A4 P08684 3/20 0.33
ALOX12 P18054 2/20 0.33
ALOX5 P09917 1/20 0.33
ALOX15 P16050 1/20 0.33
PTGS1 P23219 1/20 0.33
SLC6A2 P23975 1/20 0.33
MAPK1 P28482 1/20 0.33
HTR2B P41595 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
IDO1 P14902 2/20 0.32
CYP1A2 P05177 2/20 0.32
CYP2D6 P10635 2/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23685247 1.00 TDP1 (0.52) TDP1ALDH1A1CTSDHSD17B10TSHR
SCHEMBL22924828 0.88 HPGD (0.46) TDP1ALDH1A1CTSDTSHRPTGS2
SCHEMBL23977356 0.80 HSD17B10 (0.48) TDP1ALDH1A1CTSDHSD17B10TSHR
SCHEMBL19737269 0.72 ALDH1A1 (1.00) TDP1ALDH1A1CTSDHSD17B10TSHR
Hydrazobenzene SCHEMBL51179 0.72 ALDH1A1 (1.00) TDP1ALDH1A1CTSDHSD17B10TSHR
Hydrazobenzene SCHEMBL28199819 0.69 ALDH1A1 (0.92) TDP1ALDH1A1CTSDHSD17B10TSHR
Hydrazobenzene SCHEMBL29066354 0.65 ALDH1A1 (0.80) TDP1ALDH1A1CTSDHSD17B10TSHR
SCHEMBL21764766 0.64 ALDH1A1 (0.79) TDP1ALDH1A1CTSDHSD17B10TSHR
SCHEMBL22620524 0.63 ALDH1A1 (0.81) TDP1ALDH1A1CTSDHSD17B10TSHR
SCHEMBL30806211 0.63

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022063094-A1 TETRAHYDROISOQUINOLINE DERIVATIVE AND USE THEREOF 南京明德新药研发有限公司 2022-03-31 WO disclosed
WO-2020216240-A1 DICYCLIC ALKANE COMPOUND USEFUL AS INHIBITOR OF PLASMA KALLIKREIN 南京明德新药研发有限公司 2020-10-29 WO disclosed
WO-2020200314-A1 NITROGEN-CONTAINING SPIRO DERIVATIVE AS RET INHIBITOR 南京明德新药研发有限公司 2020-10-08 WO disclosed
WO-2020156568-A1 FLUOROVINYLBENZAMIDE COMPOUND AS PD-L1 IMMUNOMODULATOR 南京明德新药研发有限公司 2020-08-06 WO disclosed
WO-2020063855-A1 QUINOLINO-PYRROLIDIN-2-ONE DERIVATIVE AND APPLICATION THEREOF 南京明德新药研发有限公司 2020-04-02 WO disclosed