SCHEMBL22924828

SCHEMBL22924828

Cc1ccccccc(NNC2=C/C=C\C=C/C=C\C=C/C=C\2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 5/20 0.46
ALDH1A1 P00352 5/20 0.42
ALOX12 P18054 4/20 0.42
TDP1 Q9NUW8 3/20 0.42
KDM4E B2RXH2 3/20 0.42
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
GAA P10253 2/20 0.42
GFER P55789 2/20 0.42
CTSD P07339 1/20 0.40
PTGS2 P35354 1/20 0.39
LMNA P02545 2/20 0.37
TSHR P16473 1/20 0.37
ACHE P22303 1/20 0.37
HTT P42858 1/20 0.36
MAPT P10636 5/20 0.35
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21851206 0.88 TDP1 (0.52) HPGDALDH1A1ALOX12TDP1KDM4E
SCHEMBL23685247 0.88 TDP1 (0.52) HPGDALDH1A1ALOX12TDP1KDM4E
SCHEMBL21465958 0.78 HPGD (0.71) HPGDALDH1A1ALOX12TDP1KDM4E
Hydrochloric Acid SCHEMBL29106619 0.75 HPGD (0.68) HPGDALDH1A1ALOX12TDP1KDM4E
SCHEMBL23977356 0.70 HSD17B10 (0.48) HPGDALDH1A1ALOX12TDP1KDM4E
SCHEMBL2683360 0.68 TDP1 (0.57) HPGDALDH1A1ALOX12TDP1KDM4E
SCHEMBL6863517 0.66 GAA (0.57) HPGDALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL172875 0.65 HPGD (1.00) HPGDALDH1A1ALOX12TDP1CYP1A2
SCHEMBL24137168 0.65 HPGD (1.00) HPGDALDH1A1ALOX12TDP1CYP1A2
SCHEMBL9461706 0.65 HPGD (1.00) HPGDALDH1A1ALOX12TDP1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021013209-A1 MACROCYCLIC DERIVATIVES AS FACTOR XIA INHIBITORS 南京明德新药研发有限公司 2021-01-28 WO disclosed