SCHEMBL2185605

SCHEMBL2185605

Cn1cnc(-c2nc(N)c3ccncc3n2)c1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.46
ADORA1 P30542 1/20 0.46
CYP2E1 P05181 1/20 0.44
CYP2A6 P11509 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2B6 P20813 1/20 0.44
CYP2C19 P33261 1/20 0.44
MAP3K7 O43318 1/20 0.42
TAB1 Q15750 1/20 0.42
MAPT P10636 1/20 0.40
LATS1 O95835 12/20 0.39
LATS2 Q9NRM7 9/20 0.39
LRRK2 Q5S007 1/20 0.39
JAK2 O60674 1/20 0.38
JAK1 P23458 1/20 0.38
JAK3 P52333 1/20 0.38
KDM2B Q8NHM5 1/20 0.36
PHF8 Q9UPP1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17503745 0.84 CYP2E1 (0.44) ADORA2AADORA1CYP2E1CYP2A6CYP2C9
SCHEMBL2188560 0.82 ADORA1 (0.58) ADORA2AADORA1
SCHEMBL2190316 0.74 ADORA1 (0.53) ADORA2AADORA1CYP2E1CYP2A6CYP2C9
SCHEMBL21875480 0.71 LATS1 (0.61) LATS1LATS2
SCHEMBL2184224 0.71 ADORA2A (0.47) ADORA2AADORA1CYP2E1CYP2A6CYP2C9
SCHEMBL2187983 0.71 ADORA2A (0.56) ADORA2AADORA1CYP2E1CYP2A6CYP2C9
SCHEMBL15645485 0.70 LATS1 (0.65) MAPTLATS1LATS2
SCHEMBL18230128 0.69 CYP2E1 (0.53) CYP2E1CYP2A6CYP2C9CYP2B6CYP2C19
SCHEMBL2186774 0.69 ADORA2A (0.46) ADORA2AADORA1CYP2E1CYP2A6CYP2C9
SCHEMBL15644916 0.69 LATS1 (0.50) LATS1LATS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346859-A1 HETEROCYCLIC JAK KINASE INHIBITORS AstraZeneca AB (SE) 2011-07-27 EP disclosed