SCHEMBL2188560

SCHEMBL2188560

Cn1cnc(-c2nc(N)c3ccccc3n2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.58
ADORA2A P29274 1/20 0.58
CYP1A1 P04798 5/20 0.49
CYP1A2 P05177 5/20 0.49
CYP1B1 Q16678 5/20 0.49
DCPS Q96C86 1/20 0.45
HTR3A P46098 2/20 0.44
HRH4 Q9H3N8 1/20 0.44
MAOA P21397 1/20 0.44
ACHE P22303 2/20 0.41
KDM4E B2RXH2 3/20 0.40
ALDH1A1 P00352 2/20 0.40
GLA P06280 2/20 0.40
GAA P10253 2/20 0.40
HPGD P15428 2/20 0.40
HSD17B10 Q99714 2/20 0.40
ADORA3 P0DMS8 1/20 0.40
NCF1 P14598 2/20 0.40
ALOX15 P16050 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2190316 0.83 ADORA1 (0.53) ADORA1ADORA2AACHEADORA3
SCHEMBL2185605 0.82 ADORA2A (0.46) ADORA1ADORA2A
SCHEMBL2642270 0.76 CYP1A1 (0.51) ADORA1CYP1A1CYP1A2CYP1B1DCPS
SCHEMBL2184224 0.74 ADORA2A (0.47) ADORA1ADORA2AHRH4
SCHEMBL2187983 0.74 ADORA2A (0.56) ADORA1ADORA2ACYP1A2
SCHEMBL3301792 0.74 ADORA2A (1.00) ADORA1ADORA2A
SCHEMBL31169377 0.73 METAP1 (0.66) ADORA1ADORA2ACYP1A1CYP1A2CYP1B1
SCHEMBL30394017 0.73 METAP1 (0.66) ADORA1ADORA2ACYP1A1CYP1A2CYP1B1
SCHEMBL10705638 0.73 METAP1 (0.66) ADORA1ADORA2ACYP1A1CYP1A2CYP1B1
SCHEMBL11357725 0.71 CYP1A1 (0.56) CYP1A1CYP1A2CYP1B1DCPS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346859-A1 HETEROCYCLIC JAK KINASE INHIBITORS AstraZeneca AB (SE) 2011-07-27 EP disclosed