SCHEMBL21861591

SCHEMBL21861591

Brc1ccc(N2CC3CCC2C3)nc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 9/20 0.44
PDE10A Q9Y233 1/20 0.38
GRIN2D O15399 1/20 0.36
GRIN3B O60391 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2A Q12879 1/20 0.36
GRIN2B Q13224 1/20 0.36
GRIN2C Q14957 1/20 0.36
GRIN3A Q8TCU5 1/20 0.36
CHRNA7 P36544 1/20 0.36
KCNH2 Q12809 1/20 0.36
OPRM1 P35372 1/20 0.34
OPRL1 P41146 1/20 0.34
AKR1C3 P42330 1/20 0.33
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
MCHR1 Q99705 1/20 0.32
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1108634 0.81 MAP3K12 (0.44) MAP3K12PDE10AGRIN2DGRIN3BGRIN1
SCHEMBL25855693 0.81 MAP3K12 (0.50) MAP3K12GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL12879203 0.79 MAP3K12 (0.44) MAP3K12CHRNA7KCNH2ALDH1A1POLB
SCHEMBL26151688 0.78 MAP3K12 (0.42) MAP3K12CHRNA7KCNH2MCHR1
SCHEMBL25855694 0.76 MAPT (0.51) MAP3K12ALDH1A1POLBMCHR1
SCHEMBL12879195 0.75 HRH3 (0.41) MAP3K12ALDH1A1POLB
SCHEMBL4515938 0.73 CHRNA7 (0.37) PDE10AGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL21588369 0.73 ADK (0.49) MAP3K12PDE10A
SCHEMBL21588292 0.73 ADK (0.49) MAP3K12PDE10A
SCHEMBL31108110 0.73 CHRNB2 (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3193880-B1 INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL LILLY CO ELI (US) 2020-03-25 EP disclosed