SCHEMBL21864574

SCHEMBL21864574

NC(=O)c1ccc2oc(=O)cc(-c3ccc(OCC4CC4)cc3)c2c1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP15 Q460N3 4/20 0.56
PARP10 Q53GL7 4/20 0.56
PARP2 Q9UGN5 2/20 0.56
CHEK2 O96017 6/20 0.47
HPGD P15428 6/20 0.41
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 2/20 0.41
LMNA P02545 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KMT2A Q03164 3/20 0.41
HTT P42858 2/20 0.40
GPR35 Q9HC97 1/20 0.40
FFAR4 Q5NUL3 1/20 0.40
USP2 O75604 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21864570 0.85 CHEK2 (0.47) PARP10CHEK2HPGDALDH1A1KDM4E
SCHEMBL21830613 0.81 HPGD (0.37) PARP10CHEK2HPGDALDH1A1KDM4E
SCHEMBL21864586 0.78 CHEK2 (0.42) CHEK2HPGDALDH1A1KDM4ELMNA
SCHEMBL21864737 0.78 NOD2 (0.44) HPGDALDH1A1KDM4ELMNASMN1; SMN2
SCHEMBL21864581 0.78 ABL1 (0.45) CHEK2HPGDALDH1A1KDM4ELMNA
SCHEMBL21864597 0.77 KMT2A (0.44) HPGDALDH1A1KDM4ELMNASMN1; SMN2
SCHEMBL21864571 0.76 IKBKE (0.41) CHEK2HPGDALDH1A1KDM4EKMT2A
SCHEMBL10138332 0.75 PRKCZ (0.59) PARP15PARP10PARP2CHEK2
SCHEMBL21864584 0.75 CA12 (0.39) HPGDALDH1A1KDM4ELMNAKMT2A
SCHEMBL21864601 0.75 CA12 (0.40) HPGDALDH1A1KDM4ELMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020071550-A1 CDK8 INHIBITOR AND USE OF SAME 京都薬品工業株式会社 2020-04-09 WO disclosed