SCHEMBL21864629

SCHEMBL21864629

NC(=O)c1ccc2cccc(C3=CCC(OCCOC4CCOCC4)CC3)c2c1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 13/20 0.41
HTR1B P28222 4/20 0.41
HTR1E P28566 2/20 0.39
HTR1A P08908 1/20 0.39
GRM2 Q14416 1/20 0.34
CHEK2 O96017 1/20 0.33
PDE4D Q08499 1/20 0.32
SCN9A Q15858 1/20 0.32
XIAP P98170 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21864605 0.81 HTR1D (0.40) HTR1DHTR1BHTR1EHTR1AGRM2
SCHEMBL21831364 0.80 CHEK2 (0.40) CHEK2
SCHEMBL21864582 0.77 MTNR1B (0.39) HTR1DHTR1BHTR1ASCN9AXIAP
SCHEMBL21864603 0.75 HTR1D (0.46) HTR1DHTR1BHTR1EHTR1AGRM2
SCHEMBL21830577 0.71 MTNR1A (0.42)
SCHEMBL21864625 0.70 HTR1D (0.40) HTR1DHTR1BHTR1EHTR1APDE4D
SCHEMBL21831363 0.70 CHEK2 (0.38) CHEK2
SCHEMBL578566 0.69 SLC22A12 (0.41) CHEK2
SCHEMBL1318385 0.67 CDK8 (0.42) CHEK2PDE4DSCN9A
SCHEMBL21864624 0.67 HTR1D (0.38) HTR1DHTR1BHTR1EHTR1AGRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020071550-A1 CDK8 INHIBITOR AND USE OF SAME 京都薬品工業株式会社 2020-04-09 WO disclosed