SCHEMBL21869801

SCHEMBL21869801

O=C(OCc1ccc(O)cc1)[C@@H]1CCC(=O)N1Cc1ccc(F)cc1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.51
POLB P06746 1/20 0.51
KMT2A Q03164 2/20 0.49
CYP2D6 P10635 2/20 0.49
CYP2C19 P33261 2/20 0.49
MEN1 O00255 1/20 0.49
HCRTR2 O43614 3/20 0.47
TSHR P16473 2/20 0.47
ALOX15 P16050 1/20 0.47
HDAC1 Q13547 1/20 0.46
HDAC2 Q92769 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP2C9 P11712 1/20 0.46
P2RX7 Q99572 1/20 0.45
HCRTR1 O43613 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21869796 0.92 P2RX7 (0.54) GAAPOLBKMT2ACYP2D6CYP2C19
SCHEMBL28650737 0.92 P2RX7 (0.54) GAAPOLBKMT2ACYP2D6CYP2C19
SCHEMBL21869790 0.91 GAA (0.62) GAAPOLBKMT2ACYP2D6CYP2C19
SCHEMBL21869797 0.91 GAA (0.49) GAAPOLBKMT2ACYP2D6CYP2C19
SCHEMBL21869799 0.89 ITGB1 (0.52) KMT2AHDAC1HDAC2P2RX7
SCHEMBL21869800 0.89 HCRTR2 (0.52) GAAPOLBKMT2ACYP2D6CYP2C19
SCHEMBL21869753 0.88 KMT2A (0.63) GAAKMT2ACYP2C19ALDH1A1CYP2C9
SCHEMBL21869791 0.88 GAA (0.49) GAAPOLBKMT2ACYP2D6CYP2C19
SCHEMBL21869759 0.86 KMT2A (0.49) KMT2AHCRTR2HDAC1HCRTR1
SCHEMBL6997222 0.85 GAA (0.58) GAAPOLBKMT2ACYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109180552-B Substituted 5-oxo pyrrolidine derivative and preparation method and application thereof 沈阳药科大学 2021-10-26 CN disclosed
WO-2020063388-A1 SUBSTITUTED 5-OXOPYRROLIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND USE THEREOF 沈阳药科大学 2020-04-02 WO disclosed