SCHEMBL21870720

SCHEMBL21870720

CC/N=C(\N)Nc1cccc(S(C)(=O)=O)c1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1C Q13936 1/20 0.41
SCN5A Q14524 1/20 0.41
SIGMAR1 Q99720 3/20 0.36
GRIN2D O15399 2/20 0.36
GRIN3B O60391 2/20 0.36
GRIN1 Q05586 2/20 0.36
GRIN2A Q12879 2/20 0.36
GRIN2B Q13224 2/20 0.36
GRIN2C Q14957 2/20 0.36
GRIN3A Q8TCU5 2/20 0.36
CA1 P00915 5/20 0.35
CA2 P00918 5/20 0.35
CHIT1 Q13231 1/20 0.35
PSIP1 O75475 1/20 0.35
PTGIR P43119 2/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
CCR2 P41597 1/20 0.34
HTR6 P50406 1/20 0.34
CA9 Q16790 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6676349 0.77 CACNA1C (0.48) CACNA1CSCN5ASIGMAR1GRIN2DGRIN3B
SCHEMBL21870800 0.72 CCR2 (0.38) CA1CA2MEN1KMT2ACCR2
SCHEMBL23962785 0.71 HTR6 (0.46) CA1CA2PSIP1CCR2HTR6
SCHEMBL23678601 0.70 CCR2 (0.32) CA1CA2CCR2JAK2JAK1
SCHEMBL20399181 0.67 MEN1 (0.41) CA1CA2MEN1KMT2ACA9
SCHEMBL6675317 0.67 CACNA1C (0.49) CACNA1CSCN5ASIGMAR1GRIN2DGRIN3B
SCHEMBL6676424 0.66 CACNA1C (0.48) CACNA1CSCN5ASIGMAR1GRIN2DGRIN3B
Hydrochloric Acid SCHEMBL6674250 0.66 CACNA1C (0.48) CACNA1CSCN5ASIGMAR1GRIN2DGRIN3B
SCHEMBL28340525 0.66 CA1 (0.39) CA1CA2MEN1KMT2ACA9
Hydrochloric Acid SCHEMBL6675369 0.65 CACNA1C (0.47) CACNA1CSCN5ASIGMAR1GRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020057669-A1 AROMATIC HETEROCYCLIC COMPOUND WITH KINASE INHIBITORY ACTIVITY 上海轶诺药业有限公司 2020-03-26 WO disclosed