SCHEMBL2187343

SCHEMBL2187343

CCN(C(=O)c1csc(F)n1)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.49
ALDH1A1 P00352 3/20 0.49
GLA P06280 1/20 0.49
HTT P42858 1/20 0.47
TP53 P04637 1/20 0.47
HPGD P15428 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
THRA P10827 1/20 0.41
THRB P10828 1/20 0.41
ADORA2A P29274 1/20 0.40
GRM1 Q13255 1/20 0.40
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1246763 0.84 ALDH1A1 (0.50) TSHRALDH1A1GLAHTTTP53
SCHEMBL2186976 0.83 TP53 (0.54) TSHRALDH1A1GLAHTTTP53
SCHEMBL11020367 0.72 ALDH1A1 (0.53) TSHRALDH1A1GLAHTTTP53
SCHEMBL13730143 0.70 ALDH1A1 (0.52) TSHRALDH1A1GLAHTTTP53
SCHEMBL13729834 0.70 ALDH1A1 (0.52) TSHRALDH1A1GLAHTTTP53
SCHEMBL1006444 0.70 HTT (0.71) TSHRALDH1A1GLAHTTTP53
SCHEMBL3454955 0.70 TP53 (0.67) TSHRALDH1A1GLAHTTTP53
SCHEMBL3638058 0.68 ALDH1A1 (0.70) TSHRALDH1A1GLAHTTTP53
Hydrochloric Acid SCHEMBL9049882 0.68 MEN1 (0.60) TSHRALDH1A1GLAHTTTP53
SCHEMBL4111567 0.68 MEN1 (0.52) TSHRALDH1A1GLAHTTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7973061-B2 Anaplastic lymphoma kinase modulators and methods of use EXELIXIS, INC. (US) 2011-07-05 US disclosed
US-20090186905-A1 ANAPLASTIC LYMPHOMA KINASE MODULATORS AND METHODS OF USE EXELIXIS, INC. (US) 2009-07-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090186905-A1 ANAPLASTIC LYMPHOMA KINASE MODULATORS AND METHODS OF USE ALK, BCL3, MCL1 TSHR 1413/4885ALDH1A1 1466/4885GLA 3345/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.