SCHEMBL2187541

SCHEMBL2187541

C=CCOc1cc(Br)ccc1CC=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
HTT P42858 1/20 0.48
HPGD P15428 3/20 0.48
ALDH1A1 P00352 2/20 0.48
GAA P10253 1/20 0.39
TSHR P16473 1/20 0.39
LIG1 P18858 1/20 0.37
ATM Q13315 1/20 0.36
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA9 Q16790 1/20 0.35
KDM4E B2RXH2 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MAPT P10636 2/20 0.35
NPC1 O15118 1/20 0.35
TP53 P04637 1/20 0.35
RAB9A P51151 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2187712 0.88 MAPK1 (0.59) MAPK1MEN1KMT2AHTTHPGD
SCHEMBL14059336 0.81 MAPT (0.46) MAPK1HPGDALDH1A1GAATSHR
SCHEMBL21598387 0.81 TSHR (0.45) KMT2AHTTHPGDALDH1A1GAA
SCHEMBL2186993 0.81 HPGD (0.58) MAPK1MEN1KMT2AHTTHPGD
SCHEMBL4619965 0.78 HPGD (0.54) MAPK1MEN1KMT2AHTTHPGD
SCHEMBL29383173 0.77 PYCR1 (0.48) MAPK1MEN1KMT2AHTTALDH1A1
SCHEMBL1824266 0.77 PYCR1 (0.48) MAPK1MEN1KMT2AHTTALDH1A1
SCHEMBL3818208 0.77 KDM4E (0.50) MAPK1HTTHPGDALDH1A1GAA
SCHEMBL5210543 0.75 HPGD (0.58) MAPK1MEN1KMT2AHTTHPGD
SCHEMBL2219521 0.74 HPGD (0.66) MAPK1MEN1KMT2AHTTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2342179-A1 COMPOUNDS FOR INHIBITING SEMICARBAZIDE-SENSITIVE AMINE OXIDASE (SSAO) / VASCULAR ADHESION PROTEIN-1 (VAP-1) AND USES THEREOF FOR TREATMENT AND PREVENTION OF DISEASES Semmelweis Egyetem (HU) 2011-07-13 EP disclosed
WO-2010029379-A1 COMPOUNDS FOR INHIBITING SEMICARBAZIDE-SENSITIVE AMINE OXIDASE (SSAO) / VASCULAR ADHESION PROTEIN-1 (VAP-1) AND USES THEREOF FOR TREATMENT AND PREVENTION OF DISEASES SEMMELWEIS EGYETEM (HU) 2010-03-18 WO disclosed