SCHEMBL2188145

SCHEMBL2188145

CCOc1cc(CCNC(=O)c2csc(CNC(=O)COc3ccc(OC(F)(F)F)cc3)n2)ccc1OC.COc1ccccc1CNC(=O)c1csc(CNC(=O)COc2ccc(OC(F)(F)F)cc2)n1.Cc1cccc(CCNC(=O)c2csc(CNC(=O)COc3ccc(OC(F)(F)F)cc3)n2)c1.O=C(COc1ccc(OC(F)(F)F)cc1)NCc1nc(C(=O)NCC(c2ccccc2)c2ccccc2)cs1.O=C(COc1ccc(OC(F)(F)F)cc1)NCc1nc(C(=O)NCCc2cccs2)cs1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTT P42858 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
PTGER1 P34995 2/20 0.37
SMN1; SMN2 Q16637 5/20 0.36
NPC1 O15118 1/20 0.36
LMNA P02545 2/20 0.35
PKM P14618 1/20 0.35
SLC40A1 Q9NP59 1/20 0.35
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 2/20 0.34
GAA P10253 1/20 0.34
POLB P06746 1/20 0.34
TP53 P04637 1/20 0.34
PPARG P37231 1/20 0.34
PPARD Q03181 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4540788 0.97 MAPT (0.38) MAPTCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL2188149 0.88 MAPT (0.37) MAPTCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL4383985 0.82 LMNA (0.47) MAPTPTGER1SMN1; SMN2LMNAPKM
SCHEMBL12407097 0.79 TRPV1 (0.45) MAPTCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL4390910 0.77 MAPT (0.61) MAPTCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL12407087 0.76 HPGD (0.47) MAPTCYP1A2CYP3A4CYP2C19SMN1; SMN2
SCHEMBL4387708 0.75 TRPV1 (0.44) MAPTHTTSMN1; SMN2NPC1LMNA
SCHEMBL12482017 0.74 LMNA (0.49) MAPTSMN1; SMN2LMNAPKMALDH1A1
SCHEMBL4562630 0.74 SMN1; SMN2 (0.42) CYP1A2CYP3A4CYP2C9CYP2C19SMN1; SMN2
SCHEMBL4390454 0.74 MAPT (0.46) MAPTCYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7973061-B2 Anaplastic lymphoma kinase modulators and methods of use EXELIXIS, INC. (US) 2011-07-05 US claimed