SCHEMBL2188149

SCHEMBL2188149

CCOc1cc(CCc2sc(CNC(=O)COc3ccc(OC(F)(F)F)cc3)nc2C(N)=O)ccc1OC.COc1ccccc1CNC(=O)c1csc(CNC(=O)COc2ccc(OC(F)(F)F)cc2)n1.Cc1cccc(CCc2sc(CNC(=O)COc3ccc(OC(F)(F)F)cc3)nc2C(N)=O)c1.NC(=O)c1nc(CNC(=O)COc2ccc(OC(F)(F)F)cc2)sc1CC(c1ccccc1)c1ccccc1.NC(=O)c1nc(CNC(=O)COc2ccc(OC(F)(F)F)cc2)sc1CCc1cccs1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.37
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
NPC1 O15118 1/20 0.33
PPARG P37231 1/20 0.32
PPARD Q03181 1/20 0.32
PPARA Q07869 1/20 0.32
TP53 P04637 1/20 0.32
CTSD P07339 1/20 0.31
SLC40A1 Q9NP59 1/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
HCRTR2 O43614 2/20 0.31
UBE2I P63279 1/20 0.31
SAE1 Q9UBE0 1/20 0.31
UBA2 Q9UBT2 1/20 0.31
PTGER1 P34995 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2188145 0.88 MAPT (0.40) MAPTCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL4540788 0.85 MAPT (0.38) MAPTCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL4383985 0.73 LMNA (0.47) MAPTTP53SMN1; SMN2PTGER1KMT2A
SCHEMBL4390910 0.73 MAPT (0.61) MAPTCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL2188096 0.71 MAPT (0.33) MAPTCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL2189359 0.71 CNR1 (0.33) MAPTTP53
SCHEMBL12407097 0.70 TRPV1 (0.45) MAPTCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL5670152 0.70 CYP1A2 (0.50) MAPTCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL4550530 0.70 DGAT2 (0.33)
SCHEMBL2176692 0.70 MAPT (0.52) MAPTCYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7973061-B2 Anaplastic lymphoma kinase modulators and methods of use EXELIXIS, INC. (US) 2011-07-05 US claimed