SCHEMBL21882677

SCHEMBL21882677

COC(=O)C(Cc1cccnc1)Oc1cc(Cl)cc(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
NLRP3 Q96P20 1/20 0.44
NAMPT P43490 1/20 0.43
HTT P42858 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
ALDH1A1 P00352 4/20 0.42
MAPT P10636 3/20 0.41
LMNA P02545 2/20 0.41
POLB P06746 1/20 0.41
HPGD P15428 1/20 0.41
PTPN1 P18031 1/20 0.41
MAPK1 P28482 1/20 0.41
GAA P10253 1/20 0.41
CACNA1I Q9P0X4 1/20 0.41
PPARG P37231 2/20 0.40
PPARA Q07869 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
FDPS P14324 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18055529 0.86 PPARA (0.56) PPARGPPARA
SCHEMBL28171714 0.85 PPARA (0.54) PPARGPPARA
SCHEMBL19912667 0.85 PPARA (0.56) PTPN1PPARGPPARA
SCHEMBL19803711 0.85 PPARA (0.56) PTPN1PPARGPPARA
Lithium Ion SCHEMBL18039148 0.84 MEN1 (0.44) MEN1KMT2ANAMPTMAPTMAPK1
SCHEMBL23809782 0.83 HTRA1 (0.47) ALDH1A1MAPTPTPN1MAPK1PPARG
SCHEMBL19912668 0.83 HTRA1 (0.47) ALDH1A1MAPTPTPN1MAPK1PPARG
SCHEMBL11364236 0.74 PPARG (0.52) MEN1KMT2APOLBHPGDPPARG
SCHEMBL16508902 0.74 TBXAS1 (0.57) KMT2ANLRP3HTTSMN1; SMN2ALDH1A1
SCHEMBL21016946 0.73 HTRA1 (0.53) NLRP3PTPN1PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3262026-B1 NEW TRIFLUOROMETHYLPROPANAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2020-03-18 EP disclosed