SCHEMBL21884831

SCHEMBL21884831

CCOc1ccc2c(Oc3ccc4[nH]c(C)cc4c3F)ccnc2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 15/20 0.56
PDGFRB P09619 3/20 0.56
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 1/20 0.46
TSHR P16473 1/20 0.46
KMT2A Q03164 1/20 0.46
HSD17B10 Q99714 1/20 0.46
FGFR1 P11362 3/20 0.42
CYP3A4 P08684 2/20 0.42
EPHB6 O15197 2/20 0.42
RIPK2 O43353 2/20 0.42
STK10 O94804 2/20 0.42
MAP4K4 O95819 2/20 0.42
ABL1 P00519 2/20 0.42
EGFR P00533 2/20 0.42
LCK P06239 2/20 0.42
CSF1R P07333 2/20 0.42
RET P07949 2/20 0.42
HCK P08631 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30365215 0.89 KDR (0.60) KDRPDGFRBALDH1A1FGFR1CYP3A4
SCHEMBL18265407 0.84 KDR (0.56) KDRPDGFRBFGFR1CYP3A4EPHB6
SCHEMBL21884884 0.83 KDR (0.75) KDRPDGFRBFGFR1EPHB6RIPK2
SCHEMBL21806043 0.83 KDR (0.59) KDRPDGFRBFGFR1CYP3A4EPHB6
SCHEMBL21805901 0.82 KDR (0.54) KDRPDGFRBFGFR1CYP3A4EPHB6
SCHEMBL21884846 0.81 KDM4E (0.46) KDRPDGFRBKDM4EMEN1ALDH1A1
SCHEMBL21659077 0.81 KDR (0.60) KDRPDGFRBALDH1A1FGFR1EPHB6
SCHEMBL21884868 0.80 KDR (0.60) KDRPDGFRBFGFR1EPHB6RIPK2
SCHEMBL22328212 0.80 KDR (0.60) KDRPDGFRBFGFR1CYP3A4EPHB6
SCHEMBL18265416 0.80 KDR (0.77) KDRPDGFRBFGFR1EPHB6RIPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112996784-B Indole derivatives and their use in medicine 北京越之康泰生物医药科技有限公司 2023-05-30 CN disclosed
WO-2020057403-A1 INDOLE DERIVATIVE AND MEDICAL APPLICATION THEREOF 北京越之康泰生物医药科技有限公司 2020-03-26 WO disclosed