SCHEMBL21885846

SCHEMBL21885846

Cc1cc2ncc(Cl)nc2[nH]1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
CCNB2 O95067 1/20 0.39
CDK1 P06493 1/20 0.39
CCNB1 P14635 1/20 0.39
CDK5 Q00535 1/20 0.39
CDK5R1 Q15078 1/20 0.39
CCNB3 Q8WWL7 1/20 0.39
BRD4 O60885 1/20 0.33
PDE3B Q13370 3/20 0.32
PDE3A Q14432 3/20 0.32
MEN1 O00255 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PIK3CG P48736 1/20 0.32
MAP4K1 Q92918 2/20 0.31
ADORA1 P30542 2/20 0.31
ADORA2A P29274 1/20 0.31
TYRO3 Q06418 1/20 0.31
DYRK1B Q9Y463 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23443031 0.85 ALDH1A1 (0.50) ALDH1A1CDK5BRD4MEN1HTT
SCHEMBL26126300 0.80 ALDH1A1 (0.42) ALDH1A1CCNB2CDK1CCNB1CDK5
SCHEMBL13154922 0.80 CCNB2 (0.57) ALDH1A1CCNB2CDK1CCNB1CDK5
SCHEMBL31526668 0.77 CDK5 (0.44) ALDH1A1CCNB2CDK1CCNB1CDK5
SCHEMBL24323747 0.77 ALDH1A1 (0.42) ALDH1A1CCNB2CDK1CCNB1CDK5
SCHEMBL30588641 0.77 ALDH1A1 (0.42) ALDH1A1CCNB2CDK1CCNB1CDK5
SCHEMBL30588731 0.75 ALDH1A1 (0.38) ALDH1A1CCNB2CDK1CCNB1CDK5
SCHEMBL26123090 0.75 ALDH1A1 (0.38) ALDH1A1CCNB2CDK1CCNB1CDK5
SCHEMBL12437101 0.74 CCNB2 (0.37) CCNB2CDK1CCNB1CDK5CDK5R1
SCHEMBL17090692 0.74 ADORA2A (0.38) ALDH1A1CCNB2CDK1CCNB1CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020073011-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH APJ RECEPTOR ACTIVITY ANNAPURNA BIO, INC. (US) 2020-04-09 WO disclosed