SCHEMBL2190591

SCHEMBL2190591

[CH2]n1cc(C(=O)OCC)c(C(F)(F)F)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BAZ2B Q9UIF8 1/20 0.46
BAZ2A Q9UIF9 1/20 0.46
TSHR P16473 1/20 0.43
KDM4E B2RXH2 5/20 0.43
ALDH1A1 P00352 4/20 0.41
HSD17B10 Q99714 2/20 0.41
HDAC4 P56524 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
FOS P01100 2/20 0.41
JUN P05412 2/20 0.41
NFKB1 P19838 2/20 0.41
NFKB2 Q00653 2/20 0.41
RELA Q04206 2/20 0.41
CYP1A2 P05177 1/20 0.39
HTT P42858 1/20 0.39
USP2 O75604 1/20 0.39
TP53 P04637 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8871467 0.83 BAZ2B (0.47) BAZ2BBAZ2ATSHRKDM4EALDH1A1
SCHEMBL2186999 0.80 KDM4E (0.42) BAZ2BBAZ2ATSHRKDM4EALDH1A1
SCHEMBL2188450 0.79 BAZ2B (0.43) BAZ2BBAZ2ATSHRKDM4EALDH1A1
SCHEMBL2185981 0.77 KDM4E (0.53) TSHRKDM4EALDH1A1HSD17B10HDAC4
SCHEMBL10560157 0.76 KDM4E (0.42) BAZ2BBAZ2ATSHRKDM4EALDH1A1
SCHEMBL11937691 0.74 HPGD (0.43) TSHRKDM4EALDH1A1HTTHPGD
SCHEMBL1994129 0.72 TSHR (0.67) TSHRKDM4EALDH1A1HSD17B10HDAC4
SCHEMBL3979313 0.72 AR (0.38) BAZ2BBAZ2ATSHRKDM4EALDH1A1
SCHEMBL18149761 0.71 DGAT1 (0.41) BAZ2BBAZ2AKDM4EALDH1A1HSD17B10
SCHEMBL18149668 0.70 FOS (0.38) BAZ2BBAZ2ATSHRKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101538243-B Malononitrile compounds and their use SUMITOMO CHEMICAL CO 2012-05-09 CN disclosed
CN-101544606-B Malononitrile compound and use thereof SUMITOMO CHEMICAL CO 2012-02-29 CN disclosed
EP-1710234-B1 MALONONITRILE COMPOUND AND USE THEREOF SUMITOMO CHEMICAL CO (JP) 2011-07-13 EP disclosed
CN-1910147-B Malononitrile compounds and their use SUMITOMO CHEMICAL CO 2011-04-20 CN disclosed
CN-101544606-A Malononitrile compound and use thereof SUMITOMO CHEMICAL CO 2009-09-30 CN disclosed
CN-101538243-A Malononitrile compound and use thereof SUMITOMO CHEMICAL CO 2009-09-23 CN disclosed
CN-1910147-A Malononitrile compounds and their use SUMITOMO CHEMICAL CO (JP) 2007-02-07 CN disclosed
EP-1710234-A1 MALONONITRILE COMPOUND AND USE THEREOF Sumitomo Chemical Company, Limited (JP) 2006-10-11 EP disclosed