SCHEMBL21932295

SCHEMBL21932295

CN1Cc2ccc(C(=O)O)cc2N(C)C1=O

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.48
GAA P10253 1/20 0.42
ALDH1A1 P00352 1/20 0.41
MYC P01106 4/20 0.40
NR1H2 P55055 1/20 0.39
NR1H3 Q13133 1/20 0.39
BRD4 O60885 2/20 0.39
BRD2 P25440 1/20 0.39
BRD3 Q15059 1/20 0.39
TDP2 O95551 1/20 0.38
IP6K1 Q92551 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ESR1 P03372 1/20 0.37
ALOX15 P16050 1/20 0.37
PTPN7 P35236 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30343045 1.00 LMNA (0.48) LMNAGAAALDH1A1MYCNR1H2
SCHEMBL23769015 0.78 KMT2A (0.50) ALDH1A1MEN1KMT2A
SCHEMBL30204261 0.78 LMNA (0.57) LMNAGAAALDH1A1MYCNR1H2
SCHEMBL19329581 0.78 LMNA (0.57) LMNAGAAALDH1A1MYCNR1H2
SCHEMBL5987698 0.77 HSD17B10 (0.44) LMNAGAAALDH1A1BRD4BRD2
SCHEMBL3590613 0.76 LMNA (0.56) LMNAGAAALDH1A1
SCHEMBL22290464 0.76 BRD4 (0.49) LMNAALDH1A1BRD4BRD2BRD3
SCHEMBL31173196 0.76 BRD4 (0.49) LMNAALDH1A1BRD4BRD2BRD3
SCHEMBL31065615 0.76 HDAC6 (0.41) LMNAALDH1A1MEN1KMT2A
SCHEMBL21932498 0.76 HDAC6 (0.41) LMNAALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11571423-B2 Small molecule modulators of human sting CURADEV PHARMA LIMITED (GB) 2023-02-07 US disclosed
EP-3642198-B1 SMALL MOLECULE MODULATORS OF HUMAN STING CURADEV PHARMA LTD (GB) 2022-03-16 EP disclosed
US-20200147083-A1 SMALL MOLECULE MODULATORS OF HUMAN STING CURADEV PHARMA LIMITED (GB) 2020-05-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11571423-B2 Small molecule modulators of human sting STING1, IRF3, CGAS LMNA 4164/4885GAA 1176/4885ALDH1A1 4772/4885
US-20200147083-A1 SMALL MOLECULE MODULATORS OF HUMAN STING STING1, IRF3, CGAS LMNA 4164/4885GAA 1176/4885ALDH1A1 4772/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.