SCHEMBL21936036

SCHEMBL21936036

CCOC(=O)c1nc2cc(Br)ccn2c1CC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.44
PTGS2 P35354 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
MAPT P10636 1/20 0.43
PDE4A P27815 1/20 0.42
TARBP2 Q15633 1/20 0.42
ELANE P08246 3/20 0.42
ALDH1A1 P00352 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
MAPK1 P28482 1/20 0.41
KDM4E B2RXH2 3/20 0.41
GAA P10253 2/20 0.41
GLA P06280 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.40
POLB P06746 1/20 0.40
GABRA1 P14867 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21936057 0.88 MAPT (0.46) PTGS1PTGS2NPC1RAB9AMAPT
SCHEMBL31528481 0.87 RAB9A (0.52) PTGS1PTGS2NPC1RAB9AMAPT
SCHEMBL20876119 0.86 PTGS1 (0.44) PTGS1PTGS2NPC1RAB9AMAPT
SCHEMBL21937178 0.84 PTGS1 (0.42) PTGS1PTGS2NPC1RAB9AMAPT
SCHEMBL21936310 0.83 PTGDR2 (0.38) PTGS1PTGS2NPC1RAB9AALDH1A1
SCHEMBL20876131 0.83 PTGS1 (0.41) PTGS1PTGS2NPC1RAB9AMAPT
SCHEMBL20876163 0.83 PTGS1 (0.41) PTGS1PTGS2NPC1RAB9AMAPT
SCHEMBL8193697 0.80 TARBP2 (0.46) PTGS1PTGS2NPC1RAB9AMAPT
SCHEMBL31646921 0.79 ELANE (0.45) PTGS1PTGS2NPC1RAB9AMAPT
SCHEMBL1445392 0.77 NPC1 (0.56) PTGS1PTGS2NPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112601745-B Azaaryl amide derivative and preparation method and application thereof 上海和誉生物医药科技有限公司 2023-06-27 CN disclosed
CN-112601745-A Azaaryl amide derivative and preparation method and application thereof 上海和誉生物医药科技有限公司 2021-04-02 CN disclosed
WO-2020082921-A1 NITROGEN HETEROARYL AMIDE DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 上海和誉生物医药科技有限公司 2020-04-30 WO disclosed