SCHEMBL21936038

SCHEMBL21936038

CCc1c(C=O)nc2cc(C(=O)OC)ccn12

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.41
KDM4E B2RXH2 5/20 0.41
HSD17B10 Q99714 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
AKT1 P31749 1/20 0.39
AKT2 P31751 1/20 0.39
PLAU P00749 1/20 0.36
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36
TSHR P16473 1/20 0.36
HDAC1 Q13547 3/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
POLB P06746 1/20 0.35
HPGD P15428 1/20 0.35
JMJD6 Q6NYC1 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28555999 0.86 NPC1 (0.38) ALDH1A1AKT1AKT2HDAC1NPC1
SCHEMBL21936047 0.82 KDM4E (0.43) ALDH1A1KDM4EHSD17B10SMN1; SMN2AKT1
SCHEMBL21936043 0.82 KDM4E (0.43) ALDH1A1KDM4EHSD17B10SMN1; SMN2AKT1
SCHEMBL17434496 0.80 HDAC1 (0.44) ALDH1A1KDM4EHSD17B10SMN1; SMN2AKT1
SCHEMBL21936037 0.76 HDAC1 (0.34) HDAC1POLB
SCHEMBL21936499 0.75 MRGPRX4 (0.36) ALDH1A1KDM4EHSD17B10SMN1; SMN2AKT1
SCHEMBL31091944 0.75 AKT1 (0.43) ALDH1A1KDM4EHSD17B10SMN1; SMN2AKT1
SCHEMBL27272953 0.72 GRM2 (0.48) ALDH1A1KDM4EHSD17B10SMN1; SMN2AKT1
SCHEMBL976070 0.72 KDM4E (0.48) ALDH1A1KDM4EHSD17B10SMN1; SMN2AKT1
SCHEMBL24997460 0.71 ALDH1A1 (0.41) ALDH1A1KDM4EHSD17B10SMN1; SMN2AKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112601745-B Azaaryl amide derivative and preparation method and application thereof 上海和誉生物医药科技有限公司 2023-06-27 CN disclosed
WO-2020082921-A1 NITROGEN HETEROARYL AMIDE DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 上海和誉生物医药科技有限公司 2020-04-30 WO disclosed