SCHEMBL21936037

SCHEMBL21936037

CCc1c(C=O)nc2cc(Br)ccn12

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 17/20 0.34
AHR P35869 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
RECQL P46063 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21936050 0.80 KDM4E (0.38) AHRPOLBMAPTRECQL
SCHEMBL28555999 0.79 NPC1 (0.38) HDAC1POLBRECQL
SCHEMBL23726410 0.77 ALDH1A1 (0.33) AHRMAPT
SCHEMBL13144230 0.77 ALDH1A1 (0.44) MAPT
SCHEMBL21936310 0.77 PTGDR2 (0.38) HDAC1PTGDR2
SCHEMBL21937177 0.77 AHR (0.31) AHR
SCHEMBL21936038 0.76 ALDH1A1 (0.41) HDAC1POLB
SCHEMBL31528577 0.75 RAB9A (0.49) POLBMAPT
SCHEMBL21936039 0.75 HDAC1 (0.37) HDAC1AHRPTGDR2
SCHEMBL29070052 0.73 ALDH1A1 (0.43) POLBMAPTRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112601745-B Azaaryl amide derivative and preparation method and application thereof 上海和誉生物医药科技有限公司 2023-06-27 CN disclosed
CN-112601745-A Azaaryl amide derivative and preparation method and application thereof 上海和誉生物医药科技有限公司 2021-04-02 CN disclosed
WO-2020082921-A1 NITROGEN HETEROARYL AMIDE DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 上海和誉生物医药科技有限公司 2020-04-30 WO disclosed