SCHEMBL21937079

SCHEMBL21937079

c1ccc(-c2ccc(-c3ccccc3-c3cc(-c4ccccc4-c4ccc(-c5ccccn5)cc4)cc(-c4ccccc4-c4ccc(-c5cc6c(cn5)C5CCC6CC5)cc4)c3)cc2)nc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 2/20 0.36
PDK4 Q16654 1/20 0.36
KDR P35968 1/20 0.36
CHEK2 O96017 1/20 0.36
ABL1 P00519 1/20 0.36
CYP2A6 P11509 1/20 0.36
TGFBR1 P36897 6/20 0.35
BRS3 P32247 1/20 0.35
MCHR1 Q99705 1/20 0.35
CNR2 P34972 1/20 0.35
ADRA1A P35348 1/20 0.34
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP19A1 P11511 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21937205 0.92 CNR2 (0.34) ABL1CNR2
SCHEMBL21937077 0.89 FLT3 (0.35) PDK2KDRCHEK2CYP2A6TGFBR1
SCHEMBL21937001 0.83 CHEK2 (0.39) PDK2KDRCHEK2CYP2A6TGFBR1
SCHEMBL21125566 0.80 CYP2A6 (0.46) PDK2KDRCHEK2CYP2A6TGFBR1
SCHEMBL19794394 0.80 KDM4E (0.52) PDK2CHEK2CYP2A6TGFBR1CYP1A2
SCHEMBL21125828 0.78 CHEK2 (0.49) PDK2KDRCHEK2CYP2A6TGFBR1
SCHEMBL16905588 0.78 CNR2 (0.41) CNR2
SCHEMBL16905564 0.78 CNR2 (0.43) CNR2
SCHEMBL20068613 0.77 CHEK2 (0.48) PDK2KDRCHEK2CYP2A6TGFBR1
SCHEMBL25070279 0.76 TGFBR1 (0.49) PDK2KDRCYP2A6TGFBR1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020064662-A2 METHOD FOR PRODUCING STERICALLY HINDERED, NITROGEN-CONTAINING HETEROAROMATIC COMPOUNDS MERCK PATENT GMBH (DE) 2020-04-02 WO disclosed