SCHEMBL21937077

SCHEMBL21937077

c1ccc(-c2ccc(-c3ccccc3-c3cc(-c4ccccc4-c4ccc(-c5ccccn5)cc4)cc(-c4ccccc4-c4ccc(-c5cc6c(cn5)C5CC7CC(C5)CC6C7)cc4)c3)cc2)nc1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA7 P36544 1/20 0.35
CHRNA4 P43681 1/20 0.35
KDR P35968 1/20 0.34
CHEK2 O96017 1/20 0.34
TGFBR1 P36897 9/20 0.33
PDK2 Q15119 1/20 0.33
CYP2A6 P11509 1/20 0.33
CNR2 P34972 1/20 0.33
DRD2 P14416 1/20 0.32
MAPK14 Q16539 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP19A1 P11511 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21937079 0.89 PDK2 (0.36) KDRCHEK2TGFBR1PDK2CYP2A6
SCHEMBL21937205 0.80 CNR2 (0.34) CNR2
SCHEMBL21937074 0.80 NPC1 (0.39) FLT3CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL21125566 0.80 CYP2A6 (0.46) KDRCHEK2TGFBR1PDK2CYP2A6
SCHEMBL21937001 0.80 CHEK2 (0.39) KDRCHEK2TGFBR1PDK2CYP2A6
SCHEMBL16904293 0.77 CHRNB2 (0.41) FLT3CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL19794376 0.77 HSD17B1 (0.40) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL23956040 0.77 HSD17B1 (0.40) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL19794394 0.77 KDM4E (0.52) CHEK2TGFBR1PDK2CYP2A6MAPK14
SCHEMBL21125575 0.76 HSD17B1 (0.42) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020064662-A2 METHOD FOR PRODUCING STERICALLY HINDERED, NITROGEN-CONTAINING HETEROAROMATIC COMPOUNDS MERCK PATENT GMBH (DE) 2020-04-02 WO disclosed