SCHEMBL21940294

SCHEMBL21940294

Cc1cc(C#N)nnc1N1CCOC(C)C1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 9/20 0.44
STK3 Q13188 1/20 0.44
STK26 Q9P289 1/20 0.44
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
KHK P50053 1/20 0.39
FFAR2 O15552 3/20 0.35
KDM4E B2RXH2 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21940791 1.00 LRRK2 (0.44) LRRK2STK3STK26ALDH1A1HPGD
SCHEMBL21940800 0.83 KDM4E (0.44) ALDH1A1HPGDKDM4EHSD17B10
SCHEMBL21940802 0.83 KDM4E (0.44) ALDH1A1HPGDKDM4EHSD17B10
SCHEMBL21940293 0.83 KDM4E (0.44) ALDH1A1HPGDKDM4EHSD17B10
SCHEMBL21940582 0.83 KDM4E (0.44) ALDH1A1HPGDKDM4EHSD17B10
SCHEMBL21941078 0.83 KDM4E (0.38) ALDH1A1HPGDKHKFFAR2KDM4E
SCHEMBL21941085 0.82 LRRK2 (0.50) LRRK2STK3STK26ALDH1A1HPGD
SCHEMBL25361933 0.82 LRRK2 (0.40) LRRK2STK3STK26ALDH1A1HPGD
SCHEMBL31659922 0.81 LRRK2 (0.35) LRRK2STK3STK26
SCHEMBL21940600 0.78 LRRK2 (0.41) LRRK2STK3STK26FFAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3423445-B1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF FIBROSIS GALAPAGOS NV (BE) 2020-04-01 EP disclosed