SCHEMBL21948535

SCHEMBL21948535

Brc1cccnc1NC1[C@H]2COC[C@@H]12

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 2/20 0.41
AXL P30530 1/20 0.31
MAPK1 P28482 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
TYK2 P29597 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21961727 0.77 IDH1 (0.38) IDH1
SCHEMBL21948536 0.77 IDH1 (0.38) IDH1
SCHEMBL35212475 0.74 MAPK1 (0.57) MAPK1
SCHEMBL31437285 0.74 UTS2R (0.43) MAPK1
SCHEMBL26674860 0.74 UTS2R (0.43) MAPK1
SCHEMBL21948540 0.74 IDH1 (0.36) IDH1
SCHEMBL31441739 0.71 KDM4E (0.47) TDP1
SCHEMBL15206197 0.68 MERTK (0.45) AXL
SCHEMBL360202 0.65
SCHEMBL7466779 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020081508-A1 TYK2 INHIBITORS AND USES THEREOF NIMBUS LAKSHMI, INC. (US) 2020-04-23 WO disclosed